SCHEMBL15054527

SCHEMBL15054527

COc1cc(N)cc(S(N)(=O)=O)c1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR6 P50406 1/20 0.50
PTGS2 P35354 5/20 0.46
CA1 P00915 9/20 0.45
CA2 P00918 9/20 0.45
CA9 Q16790 8/20 0.45
CA12 O43570 4/20 0.45
CA4 P22748 2/20 0.45
CA14 Q9ULX7 2/20 0.45
CA3 P07451 1/20 0.43
APEX1 P27695 1/20 0.43
CYP2C19 P33261 1/20 0.43
ALDH1A1 P00352 2/20 0.42
CYP3A4 P08684 1/20 0.42
USP2 O75604 1/20 0.41
TSHR P16473 1/20 0.41
CA6 P23280 1/20 0.41
CA5A P35218 1/20 0.41
CA7 P43166 1/20 0.41
CA13 Q8N1Q1 1/20 0.41
TDP1 Q9NUW8 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30452587 0.89 PTGS2 (0.53) PTGS2CA1CA2CA9CA12
SCHEMBL2437487 0.83 HTR6 (0.50) HTR6PTGS2ALDH1A1CYP3A4TDP1
SCHEMBL1606727 0.82 HTR6 (0.49) HTR6CYP2C19ALDH1A1CYP3A4TSHR
SCHEMBL20241363 0.81 CA1 (0.58) CA1CA2CA9CA12CA4
SCHEMBL12325146 0.80 HTR6 (0.47) HTR6ALDH1A1CYP3A4TDP1
SCHEMBL30365875 0.79 ALDH1A1 (0.65) HTR6CA1CA2CA9CA12
SCHEMBL1804382 0.79 CA2 (0.58) CA1CA2CA9CA12CA4
SCHEMBL1172281 0.79 CA2 (0.58) CA1CA2CA9CA12CA4
SCHEMBL16829089 0.79 MAPT (0.47) HTR6ALDH1A1CYP3A4TSHR
SCHEMBL23413661 0.77 PTGS2 (0.51) PTGS2CA1CA2CA9CA12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013096151-A1 CHEMICAL COMPOUNDS GLAXOSMITHKLINE LLC (US) 2013-06-27 WO disclosed
WO-2013096153-A1 CHEMICAL COMPOUNDS GLAXOSMITHKLINE LLC (US) 2013-06-27 WO disclosed