SCHEMBL2437487

SCHEMBL2437487

COc1cc(N)cc(S(C)(=O)=O)c1

nearest known ligand 0.50

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
HTR6 P50406 1/20 0.50
ALDH1A1 P00352 2/20 0.42
CYP3A4 P08684 1/20 0.42
CYP19A1 P11511 1/20 0.40
NQO2 P16083 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
XDH P47989 2/20 0.40
PKM P14618 2/20 0.39
PTGS2 P35354 3/20 0.39
PTGS1 P23219 2/20 0.39
MAPK1 P28482 1/20 0.38
TDP1 Q9NUW8 1/20 0.38
EGFR P00533 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15054527 0.83 HTR6 (0.50) HTR6ALDH1A1CYP3A4PTGS2PTGS1
SCHEMBL1172197 0.82 L3MBTL1 (0.46) HTR6ALDH1A1CYP3A4SMN1; SMN2PTGS2
SCHEMBL2651077 0.82 G6PD (0.43) HTR6ALDH1A1CYP3A4PTGS2TDP1
SCHEMBL1606727 0.82 HTR6 (0.49) HTR6ALDH1A1CYP3A4CYP19A1NQO2
SCHEMBL31738331 0.81 HTR6 (0.45) HTR6ALDH1A1CYP3A4CYP19A1NQO2
SCHEMBL2436557 0.81 LOX (0.51) HTR6ALDH1A1CYP3A4SMN1; SMN2PKM
SCHEMBL12325146 0.80 HTR6 (0.47) HTR6ALDH1A1CYP3A4CYP19A1NQO2
SCHEMBL14633653 0.80 LOX (0.37) HTR6ALDH1A1SMN1; SMN2
SCHEMBL30365875 0.79 ALDH1A1 (0.65) HTR6ALDH1A1CYP3A4CYP19A1NQO2
SCHEMBL17263616 0.79 RAPGEF4 (0.44) ALDH1A1SMN1; SMN2XDHPKMPTGS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 125 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113045476-B Monosubstituted or disubstituted indole derivatives as dengue virus replication inhibitors 杨森制药公司 2024-07-16 CN claimed
CN-117616010-A Process for preparing (S) -2- (4-chloro-2-methoxyphenyl) -2- ((3-methoxy-5- (methylsulfonyl) phenyl) amino) -1- (1H-indol-3-yl) ketene derivatives 杨森制药公司 2024-02-27 CN claimed
CN-111303000-B Monosubstituted or disubstituted indole derivatives as dengue virus replication inhibitors 杨森制药公司 2023-11-28 CN claimed
EP-3896072-B1 MONO- OR DI-SUBSTITUTED INDOLE DERIVATIVES AS DENGUE VIRAL REPLICATION INHIBITORS JANSSEN PHARMACEUTICALS INC (US) 2022-11-16 EP claimed
EP-3350162-B1 MONO- OR DI-SUBSTITUTED INDOLE DERIVATIVES AS DENGUE VIRAL REPLICATION INHIBITORS JANSSEN PHARMACEUTICALS INC (US) 2021-07-14 EP claimed
EP-4363403-B1 PROCESSES FOR THE PREPARATION OF (S)-2-(4-CHLORO-2-METHOXYPHENYL)-2-((3-METHOXY-5-(METHYLSULFONYL)PHENYL)AMINO)-1-(1H-INDOL-3-YL)ETHENONE DERIVATIVES UNIV LEUVEN KATH (BE) 2026-05-27 EP disclosed
EP-4240331-B1 SOLID FORMULATION UNIV LEUVEN KATH (BE) 2026-04-29 EP disclosed
US-20250281457-A1 TREATMENT OR PREVENTION OF DENGUE VIRAL INFECTION KATHOLIEKE UNIVERSITEIT LEUVEN (BE) 2025-09-11 US disclosed
US-20250230127-A1 MONO- OR DI-SUBSTITUTED INDOLE DERIVATIVES AS DENGUE VIRAL REPLICATION INHIBITORS JANSSEN PHARMACEUTICALS INC (US) 2025-07-17 US disclosed
US-20250177391-A1 INHIBITORS OF DDR1 AND DDR2 FOR THE TREATMENT OF ARTHRITIS PRESIDENT AND FELLOWS OF HARVARD COLLEGE (US) 2025-06-05 US disclosed
EP-4522163-A1 TREATMENT OR PREVENTION OF DENGUE VIRAL INFECTION Janssen Pharmaceuticals, Inc. (US) 2025-03-19 EP disclosed
EP-4482825-A2 INHIBITORS OF DDR1 AND DDR2 FOR THE TREATMENT OF ARTHRITIS President and Fellows of Harvard College (US) 2025-01-01 EP disclosed
WO-2010038081-A2 HETEROCYCLIC DERIVATIVES AND METHODS OF USE THEREOF ASTRAZENECA AB (SE) 2010-04-08 WO disclosed
WO-2010038081-A2 HETEROCYCLIC DERIVATIVES AND METHODS OF USE THEREOF ASTRAZENECA AB (SE) 2010-04-08 WO disclosed
EP-2114945-A1 PTERIDINONE DERIVATIVES AS PI3-KINASES INHIBITORS Boehringer Ingelheim International GmbH (DE) 2009-11-11 EP disclosed
WO-2009109483-A1 LEUKOTRIENE B4 INHIBITORS F. HOFFMANN-LA ROCHE AG (CH) 2009-09-11 WO disclosed
US-20090227603-A1 LEUKOTRIENE B4 INHIBITORS DOMINIQUE ROMYR 2009-09-10 US disclosed
US-20090227603-A1 LEUKOTRIENE B4 INHIBITORS DOMINIQUE ROMYR 2009-09-10 US disclosed
WO-2008092831-A1 PTERIDINONE DERIVATIVES AS PI3-KINASES INHIBITORS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2008-08-07 WO disclosed
EP-1953163-A1 Pteridinone derivatives as PI3-kinases inhibitors Boehringer Ingelheim Pharma GmbH & Co. KG (DE) 2008-08-06 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090227603-A1 LEUKOTRIENE B4 INHIBITORS LTB4R2, LTB4R, LTC4S HTR6 2030/4885ALDH1A1 685/4885CYP3A4 402/4885
US-20250177391-A1 INHIBITORS OF DDR1 AND DDR2 FOR THE TREATMENT OF ARTHRITIS DDR2, DDR1, DDRGK1 HTR6 3335/4885ALDH1A1 2720/4885CYP3A4 4399/4885
US-20250281457-A1 TREATMENT OR PREVENTION OF DENGUE VIRAL INFECTION F3, FOXO3, FOXO1 HTR6 2712/4885ALDH1A1 1363/4885CYP3A4 76/4885
US-20250230127-A1 MONO- OR DI-SUBSTITUTED INDOLE DERIVATIVES AS DENGUE VIRAL REPLICATION INHIBITORS IDO1, IDO2, IRF3 HTR6 321/4885ALDH1A1 2351/4885CYP3A4 909/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.