Metiazinic Acid

Metiazinic Acid

SCHEMBL150554

CN1c2ccccc2Sc2ccc(CC(=O)O)cc21

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 4/20 0.59
NOX1 Q9Y5S8 4/20 0.59
L3MBTL1 Q9Y468 2/20 0.59
MAPT P10636 2/20 0.59
MAPK1 P28482 1/20 0.59
TDP1 Q9NUW8 1/20 0.59
MAOA P21397 1/20 0.54
BCHE P06276 4/20 0.51
HRH1 P35367 3/20 0.51
ADRA1A P35348 2/20 0.51
ADRA1D P25100 1/20 0.51
ADRA1B P35368 1/20 0.51
MEN1 O00255 2/20 0.50
KMT2A Q03164 2/20 0.50
HTR2C P28335 2/20 0.49
HTR2B P41595 2/20 0.49
HTR6 P50406 1/20 0.49
SLC6A3 Q01959 1/20 0.49
ACHE P22303 2/20 0.49
ADRA2A P08913 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Metiazinic Acid SCHEMBL10820947 1.00 LMNA (0.59) LMNANOX1L3MBTL1MAPTMAPK1
Metiazinic Acid SCHEMBL30190433 1.00 LMNA (0.59) LMNANOX1L3MBTL1MAPTMAPK1
Metiazinic Acid SCHEMBL30697757 1.00 LMNA (0.59) LMNANOX1L3MBTL1MAPTMAPK1
SCHEMBL28555924 0.86 NOX1 (0.57) LMNANOX1L3MBTL1MAPTMAPK1
SCHEMBL2669592 0.86 MAOA (0.54) LMNANOX1L3MBTL1MAPTMAPK1
SCHEMBL6850282 0.85 MAPT (0.56) LMNANOX1L3MBTL1MAPTMAPK1
SCHEMBL13295825 0.83 BCHE (0.53) LMNANOX1L3MBTL1MAPTMAPK1
SCHEMBL15101212 0.82 MAPT (0.52) LMNANOX1L3MBTL1MAPTMAPK1
Metiazinic Acid SCHEMBL7627349 0.81 LMNA (0.54) LMNANOX1L3MBTL1MAPTMAPK1
Metiazinic Acid SCHEMBL8208232 0.81 MAPT (0.56) LMNANOX1L3MBTL1MAPTMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 3381 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4628080-A1 PHARMACEUTICAL COMPOSITION FOR PREVENTION OR TREATMENT OF DRUG-RELATED PEPTIC ULCER COMPRISING ZASTAPRAZAN OR PHARMACEUTICALLY ACCEPTABLE SALT THEREOF Jeil Pharmaceutical Co., Ltd. (KR) 2025-10-08 EP claimed
EP-4470565-A1 METHOD FOR PREVENTING OR TREATING DISEASE OR DISORDER ASSOCIATED WITH ANTINEOPLASTIC AGENT OnQuality Pharmaceuticals China Ltd. (CN) 2024-12-04 EP claimed
CN-118742325-A Methods for preventing or treating diseases or conditions associated with antineoplastic agents 上海岸阔医药科技有限公司 2024-10-01 CN claimed
WO-2024117797-A1 PHARMACEUTICAL COMPOSITION FOR PREVENTION OR TREATMENT OF DRUG-RELATED PEPTIC ULCER COMPRISING ZASTAPRAZAN OR PHARMACEUTICALLY ACCEPTABLE SALT THEREOF 제일약품 주식회사 2024-06-06 WO claimed
WO-2024105529-A1 CHEMICAL DISBUDDING OF LIVESTOCK MASSEY UNIVERSITY (NZ) 2024-05-23 WO claimed
US-20240041935-A1 PREVENTION AND TREATMENT OF REPRODUCTIVE FAILURE BY REGENERATIVE CELLS AND ADJUVANTS CREATIVE MEDICAL TECHNOLOGIES, INC. (US) 2024-02-08 US claimed
EP-3752201-B1 SUSPENSION OF NANOSCALE, ORGANIC PARTICLES AND PROCESS FOR PRODUCTION THEREOF UNIV FRIEDRICH ALEXANDER ER (DE) 2023-11-22 EP claimed
WO-2023142996-A1 METHOD FOR PREVENTING OR TREATING DISEASE OR DISORDER ASSOCIATED WITH ANTINEOPLASTIC AGENT 上海岸阔医药科技有限公司 2023-08-03 WO claimed
EP-4034087-A1 LIPID VESICLE COMPOSITIONS WITH PENETRATION ENHANCING AGENTS DDS Research Inc. (CA) 2022-08-03 EP claimed
US-20220218611-A1 LIPID VESICLE COMPOSITIONS WITH PENETRATION ENHANCING AGENTS DDS RESEARCH INC. (CA) 2022-07-14 US claimed
EP-0569411-B1 ACYLAMINO-ALKYLIDEN-HYDROXY-BISPHOSPHONIC ACIDS USEFUL IN THE THERAPY OF OSTEOARTICULAR DISEASES GENTILI IST SPA (IT) 1995-03-29 EP claimed
US-5330981-A Antiinflammatory agents ISTITUTO GENTILI S.P.A. (IT) 1994-07-19 US claimed
EP-0569411-A1 ACYLAMINO-ALKYLIDEN-HYDROXY-BISPHOSPHONIC ACIDS USEFUL IN THE THERAPY OF OSTEOARTICULAR DISEASES. GENTILI IST SPA (IT) 1993-11-18 EP claimed
EP-0537313-A1 ARYLALKYL ESTERS OF 4,5-DIHYDROXY-9,10-DIHYDRO-9,10-DIOXO-2-ANTHRACENECARBOXYLIC ACID HAVING THERAPEUTICAL ACTIVITY. GENTILI IST SPA (IT) 1993-04-21 EP claimed
WO-1992019584-A1 ARYLALKYL ESTERS OF 4,5-DIHYDROXY-9,10-DIHYDRO-9,10-DIOXO-2-ANTHRACENECARBOXYLIC ACID HAVING THERAPEUTICAL ACTIVITY ISTITUTO GENTILI S.P.A. (IT) 1992-11-12 WO claimed
WO-1992013864-A1 ACYLAMINO-ALKYLIDEN-HYDROXY-BISPHOSPHONIC ACIDS USEFUL IN THE THERAPY OF OSTEOARTICULAR DISEASES ISTITUTO GENTILI S.P.A. (IT) 1992-08-20 WO claimed
EP-0040899-B1 METHOD OF DELIVERING DRUG WITH AID OF EFFERVESCENT ACTIVITY GENERATED IN ENVIRONMENT OF USE ALZA CORPORATION (US) 1984-09-12 EP claimed
EP-0072462-A2 Pharmaceutical preparations Toko Yakuhin Industry Co., Ltd. (JP) 1983-02-23 EP claimed
US-4344929-A Method of delivering drug with aid of effervescent activity generated in environment of use ALZA CORPORATION (US) 1982-08-17 US claimed
EP-0040899-A2 Method of delivering drug with aid of effervescent activity generated in environment of use ALZA CORPORATION (US) 1981-12-02 EP claimed