SCHEMBL15062024

SCHEMBL15062024

Cc1ccccc1CN1CCC(O)(C(F)(F)F)CC1

nearest known ligand 0.55

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ACHE P22303 1/20 0.55
ALDH1A1 P00352 6/20 0.54
KDM4E B2RXH2 5/20 0.54
GAA P10253 2/20 0.54
TDP1 Q9NUW8 2/20 0.54
ATM Q13315 1/20 0.54
NPSR1 Q6W5P4 1/20 0.54
KMT2A Q03164 3/20 0.54
CYP2A13 Q16696 1/20 0.53
LMNA P02545 3/20 0.51
MEN1 O00255 2/20 0.45
L3MBTL1 Q9Y468 1/20 0.44
GBA1 P04062 1/20 0.44
UBE2M P61081 1/20 0.43
DCUN1D1 Q96GG9 1/20 0.43
CCR5 P51681 1/20 0.43
MAPT P10636 1/20 0.42
HTT P42858 1/20 0.42
CXCR4 P61073 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17955425 0.83 KDM4E (0.47) ALDH1A1KDM4EGAATDP1ATM
SCHEMBL4484154 0.78 OPRL1 (0.61) ALDH1A1KDM4EGAAATMKMT2A
SCHEMBL11889011 0.77 ALDH1A1 (0.54) ACHEALDH1A1KDM4EGAATDP1
SCHEMBL329437 0.73 KMT2A (0.72) ACHEALDH1A1KDM4EGAATDP1
SCHEMBL11889055 0.72 ALDH1A1 (0.53) ACHEALDH1A1KDM4EGAATDP1
Hydrochloric Acid SCHEMBL23850614 0.72 LMNA (0.71) ACHEALDH1A1KDM4EGAATDP1
SCHEMBL1882777 0.72 KMT2A (0.70) ACHEALDH1A1KDM4EGAATDP1
SCHEMBL1164984 0.72 KMT2A (0.70) ACHEALDH1A1KDM4EGAATDP1
SCHEMBL12856255 0.72 KMT2A (0.76) ACHEALDH1A1KDM4EGAATDP1
SCHEMBL12013922 0.71 ACHE (1.00) ACHEALDH1A1KDM4EKMT2ACYP2A13

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013091773-A1 TETRAAZA-CYCLOPENTA[A]INDENYL AND THEIR USE AS POSITIVE ALLOSTERIC MODULATORS MERCK PATENT GMBH (DE) 2013-06-27 WO disclosed
EP-2607364-A1 Tetraaza-cyclopenta[a]indenyl and their use as positive allosteric modulators Ares Trading S.A. (CH) 2013-06-26 EP disclosed