SCHEMBL15062940

SCHEMBL15062940

CC#C[C@H](N[C@@H](CS(=O)(=O)CC1CC1)C(=O)NC1(C#N)CC1)C(F)(F)Oc1ccc(S(C)(=O)=O)cc1

nearest known ligand 0.57

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
CTSS P25774 18/20 0.57
CTSK P43235 16/20 0.57
CTSB P07858 15/20 0.57
CTSL P07711 15/20 0.57
CTSV O60911 1/20 0.46
CTSF Q9UBX1 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15062941 1.00 CTSS (0.57) CTSSCTSKCTSBCTSLCTSV
SCHEMBL2343904 0.88 CTSK (0.50) CTSSCTSKCTSBCTSLCTSV
SCHEMBL2442319 0.85 CTSS (0.74) CTSSCTSKCTSBCTSLCTSV
SCHEMBL2442314 0.85 CTSS (0.74) CTSSCTSKCTSBCTSLCTSV
SCHEMBL15062922 0.84 CTSS (0.45) CTSSCTSKCTSBCTSLCTSV
SCHEMBL15062923 0.84 CTSS (0.45) CTSSCTSKCTSBCTSLCTSV
SCHEMBL2398489 0.79 CTSS (0.82) CTSSCTSKCTSBCTSL
SCHEMBL2398486 0.79 CTSS (0.82) CTSSCTSKCTSBCTSL
SCHEMBL15766822 0.78 CTSS (0.47) CTSSCTSKCTSBCTSL
SCHEMBL15062901 0.76 CTSL (0.43) CTSSCTSKCTSBCTSL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2361243-B9 HALOALKYL CONTAINING COMPOUNDS AS CYSTEINE PROTEASE INHIBITORS VIROBAY INC (US) 2014-06-11 EP claimed
EP-2361243-B1 HALOALKYL CONTAINING COMPOUNDS AS CYSTEINE PROTEASE INHIBITORS VIROBAY INC (US) 2013-07-03 EP claimed
EP-2361243-B9 HALOALKYL CONTAINING COMPOUNDS AS CYSTEINE PROTEASE INHIBITORS VIROBAY INC (US) 2014-06-11 EP disclosed
EP-2361243-B1 HALOALKYL CONTAINING COMPOUNDS AS CYSTEINE PROTEASE INHIBITORS VIROBAY INC (US) 2013-07-03 EP disclosed