SCHEMBL1507919

SCHEMBL1507919

O=S(=O)(Nc1cccc2cccnc12)c1cccc2cccnc12

nearest known ligand 0.76

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC40A1 Q9NP59 15/20 0.76
TDP1 Q9NUW8 4/20 0.76
MEN1 O00255 3/20 0.76
KMT2A Q03164 3/20 0.76
NFKBIA P25963 3/20 0.76
RELA Q04206 2/20 0.76
GAA P10253 1/20 0.76
MMP2 P08253 1/20 0.71
ALDH1A1 P00352 1/20 0.71
POLB P06746 1/20 0.71
GLO1 Q04760 2/20 0.70
G6PD P11413 1/20 0.70
AGTR1 P30556 1/20 0.70
METAP2 P50579 1/20 0.70
METAP1 P53582 1/20 0.70
PAX8 Q06710 1/20 0.70
ATM Q13315 1/20 0.70
MDM4 O15151 1/20 0.69
OPRK1 P41145 1/20 0.69
MDM2 Q00987 1/20 0.69

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30854809 1.00 SLC40A1 (0.76) SLC40A1TDP1MEN1KMT2ANFKBIA
SCHEMBL27214283 0.89 SLC40A1 (0.80) SLC40A1TDP1MEN1KMT2ANFKBIA
SCHEMBL30925525 0.89 SLC40A1 (0.80) SLC40A1TDP1MEN1KMT2ANFKBIA
SCHEMBL6981201 0.88 SLC40A1 (0.73) SLC40A1TDP1MEN1KMT2ANFKBIA
SCHEMBL30925552 0.88 SLC40A1 (0.78) SLC40A1TDP1MEN1KMT2ANFKBIA
SCHEMBL27214248 0.88 SLC40A1 (0.78) SLC40A1TDP1MEN1KMT2ANFKBIA
SCHEMBL29255667 0.87 SLC40A1 (0.72) SLC40A1TDP1MEN1KMT2ANFKBIA
SCHEMBL29255668 0.87 SLC40A1 (0.68) SLC40A1TDP1MEN1KMT2ANFKBIA
SCHEMBL30854820 0.87 SLC40A1 (0.68) SLC40A1TDP1MEN1KMT2ANFKBIA
SCHEMBL30854816 0.87 SLC40A1 (0.72) SLC40A1TDP1MEN1KMT2ANFKBIA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 17 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117865886-B N- (quinoline-8-yl) quinoline-8-sulfonamide compound and application thereof 中国药科大学 2024-05-10 CN claimed
CN-117865886-A N- (quinoline-8-yl) quinoline-8-sulfonamide compound and application thereof 中国药科大学 2024-04-12 CN claimed
US-20090227626-A1 NOVEL POLYQUINOLINE DERIVATIVES AND THERAPEUTIC USE THEREOF PALUMED S.A. (FR) 2009-09-10 US claimed
CN-117865886-B N- (quinoline-8-yl) quinoline-8-sulfonamide compound and application thereof 中国药科大学 2024-05-10 CN disclosed
CN-117865886-B N- (quinoline-8-yl) quinoline-8-sulfonamide compound and application thereof 中国药科大学 2024-05-10 CN disclosed
CN-117865886-B N- (quinoline-8-yl) quinoline-8-sulfonamide compound and application thereof 中国药科大学 2024-05-10 CN disclosed
CN-117865886-A N- (quinoline-8-yl) quinoline-8-sulfonamide compound and application thereof 中国药科大学 2024-04-12 CN disclosed
CN-117865886-A N- (quinoline-8-yl) quinoline-8-sulfonamide compound and application thereof 中国药科大学 2024-04-12 CN disclosed
CN-117865886-A N- (quinoline-8-yl) quinoline-8-sulfonamide compound and application thereof 中国药科大学 2024-04-12 CN disclosed
US-8324196-B2 Polyquinoline derivatives and the therapeutic use thereof PALUMED S.A. (FR) 2012-12-04 US disclosed
US-20120277265-A1 NOVEL POLYQUINOLINE DERIVATIVES AND THE THERAPEUTIC USE THEREOF CENTRE NATIONAL DE LA RECHERCHE SCIENTIFIQUE (C.N.R.S.) (FR) 2012-11-01 US disclosed
US-8247396-B2 Polyquinoline derivatives and therapeutic use thereof PALUMED S.A. (FR) 2012-08-21 US disclosed
EP-2289891-A2 Novel polyquinoline derivates and the therapeutic use thereof Palumed S.A. (FR) 2011-03-02 EP disclosed
EP-2289891-A2 Novel polyquinoline derivates and the therapeutic use thereof Palumed S.A. (FR) 2011-03-02 EP disclosed
US-20100041653-A1 COMPOSITION AND METHODS FOR THE DESIGN AND DEVELOPMENT OF METALLO-ENZYME INHIBITORS BURNHAM INSTITUTE FOR MEDICAL RESEARCH (US) 2010-02-18 US disclosed
US-20100041653-A1 COMPOSITION AND METHODS FOR THE DESIGN AND DEVELOPMENT OF METALLO-ENZYME INHIBITORS BURNHAM INSTITUTE FOR MEDICAL RESEARCH (US) 2010-02-18 US disclosed
US-20090227626-A1 NOVEL POLYQUINOLINE DERIVATIVES AND THERAPEUTIC USE THEREOF PALUMED S.A. (FR) 2009-09-10 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120277265-A1 NOVEL POLYQUINOLINE DERIVATIVES AND THE THERAPEUTIC USE THEREOF HTT, APP, PSEN1 SLC40A1 124/4885TDP1 616/4885MEN1 1196/4885
US-20090227626-A1 NOVEL POLYQUINOLINE DERIVATIVES AND THERAPEUTIC USE THEREOF HTT, UBQLN2, UBQLN1 SLC40A1 2081/4885TDP1 860/4885MEN1 1574/4885
US-20100041653-A1 COMPOSITION AND METHODS FOR THE DESIGN AND DEVELOPMENT OF METALLO-ENZYME INHIBITORS HELZ, MMEL1, GAA SLC40A1 408/4885TDP1 1854/4885MEN1 3212/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.