SCHEMBL1508095

SCHEMBL1508095

CCOP(=O)(O)C(c1ccc(F)cc1)(c1ccc(F)cc1)c1ccccn1

nearest known ligand 0.40

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
HDAC6 Q9UBN7 5/20 0.40
ALDH1A1 P00352 2/20 0.39
CETP P11597 1/20 0.39
RAB9A P51151 2/20 0.38
NPC1 O15118 1/20 0.38
AGTR1 P30556 1/20 0.38
AHR P35869 1/20 0.37
MEN1 O00255 1/20 0.37
KMT2A Q03164 1/20 0.37
FDPS P14324 1/20 0.36
KDM4E B2RXH2 1/20 0.36
BLM P54132 1/20 0.35
CYP2D6 P10635 1/20 0.35
PTGS1 P23219 1/20 0.34
PTGS2 P35354 1/20 0.34
CHRM2 P08172 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12834657 0.86 HDAC6 (0.42) HDAC6CETPRAB9ANPC1AGTR1
SCHEMBL1507955 0.82 ALDH1A1 (0.42) ALDH1A1RAB9AMEN1KMT2AKDM4E
SCHEMBL1508012 0.78 KCNN4 (0.47) ALDH1A1MEN1KMT2AKDM4E
SCHEMBL1508091 0.78 HDAC6 (0.41) HDAC6CETPRAB9ANPC1AGTR1
SCHEMBL1507922 0.77 ALOX15 (0.38) ALDH1A1RAB9ANPC1MEN1KMT2A
SCHEMBL1508255 0.76 KMT2A (0.42) ALDH1A1NPC1MEN1KMT2AKDM4E
SCHEMBL1508218 0.75 KCNN4 (0.47) HDAC6ALDH1A1MEN1KMT2AKDM4E
SCHEMBL1508149 0.72 KCNN4 (0.41) ALDH1A1RAB9AMEN1KMT2AKDM4E
SCHEMBL8167421 0.69 FDPS (0.66) ALDH1A1MEN1KMT2AFDPSKDM4E
SCHEMBL1508245 0.69 ALDH1A1 (0.42) ALDH1A1MEN1KMT2AKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 14 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2292595-A1 Potassium channel modulators NeuroSearch AS (DK) 2011-03-09 EP claimed
EP-1911740-A1 POTASSIUM CHANNEL MODULATORS NeuroSearch A/S (DK) 2008-04-16 EP claimed
US-20070161607-A1 Potassium channel modulators SANIONA A/S (DK) 2007-07-12 US claimed
US-20050009816-A1 Potassium channel modulators SANIONA A/S (DK) 2005-01-13 US claimed
EP-1465863-A1 POTASSIUM CHANNEL MODULATORS Poseidon Pharmaceuticals A/S (DK) 2004-10-13 EP claimed
WO-2003059873-A1 POTASSIUM CHANNEL MODULATORS POSEIDON PHARMACEUTICALS A/S (DK) 2003-07-24 WO claimed
EP-2292595-A1 Potassium channel modulators NeuroSearch AS (DK) 2011-03-09 EP disclosed
US-7429618-B2 Potassium channel modulators NEUROSEARCH A/S (DK) 2008-09-30 US disclosed
EP-1911740-A1 POTASSIUM CHANNEL MODULATORS NeuroSearch A/S (DK) 2008-04-16 EP disclosed
US-20070161607-A1 Potassium channel modulators SANIONA A/S (DK) 2007-07-12 US disclosed
US-7208527-B2 Potassium channel modulators POSEIDON PHARMACEUTICALS A/S (DK) 2007-04-24 US disclosed
US-20050009816-A1 Potassium channel modulators SANIONA A/S (DK) 2005-01-13 US disclosed
EP-1465863-A1 POTASSIUM CHANNEL MODULATORS Poseidon Pharmaceuticals A/S (DK) 2004-10-13 EP disclosed
WO-2003059873-A1 POTASSIUM CHANNEL MODULATORS POSEIDON PHARMACEUTICALS A/S (DK) 2003-07-24 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050009816-A1 Potassium channel modulators KCNC1, KCNQ1, KCNA1 HDAC6 1233/4885ALDH1A1 3877/4885CETP 2344/4885
US-20070161607-A1 Potassium channel modulators KCNC1, KCNQ1, KCNA1 HDAC6 1233/4885ALDH1A1 3877/4885CETP 2344/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.