SCHEMBL15211548

SCHEMBL15211548

CC(=O)Oc1csc2cc(C=O)ccc12

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 1/20 0.40
JUN P05412 1/20 0.38
NFKB1 P19838 1/20 0.38
VCP P55072 1/20 0.37
ALDH1A1 P00352 6/20 0.37
AOX1 Q06278 1/20 0.37
TRIM24 O15164 1/20 0.37
HPGD P15428 1/20 0.37
ALDH5A1 P51649 1/20 0.37
ABAT P80404 1/20 0.37
TDP1 Q9NUW8 1/20 0.37
TRIM33 Q9UPN9 1/20 0.37
FNTA P49354 1/20 0.37
FNTB P49356 1/20 0.37
TSHR P16473 2/20 0.37
KDM4E B2RXH2 3/20 0.36
MAPT P10636 2/20 0.36
MEN1 O00255 1/20 0.36
LMNA P02545 1/20 0.36
TTR P02766 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15211511 0.80 CYP3A4 (0.41) ESR1ALDH1A1HPGDTDP1TSHR
SCHEMBL15211105 0.77 KMT2A (0.37) ESR1JUNNFKB1VCPALDH1A1
SCHEMBL15211467 0.77 KMT2A (0.37) ESR1JUNNFKB1VCPALDH1A1
SCHEMBL15211106 0.77 KMT2A (0.37) ESR1JUNNFKB1VCPALDH1A1
SCHEMBL2025468 0.74 PKM (0.51) ESR1ALDH1A1HPGDTDP1TSHR
SCHEMBL31190039 0.74 JUN (0.57) JUNNFKB1VCPALDH1A1AOX1
SCHEMBL320559 0.74 JUN (0.57) JUNNFKB1VCPALDH1A1AOX1
SCHEMBL16693081 0.73 CYP2A6 (0.42) ALDH1A1AOX1TRIM24HPGDALDH5A1
SCHEMBL15211611 0.72 CYP3A4 (0.40) ESR1NFKB1ALDH1A1TSHRKDM4E
SCHEMBL28073642 0.72 ALOX15 (0.40) ESR1VCPALDH1A1KDM4EMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2838891-A1 AROMATIC RING COMPOUND Takeda Pharmaceutical Company Limited (JP) 2015-02-25 EP disclosed
WO-2013125732-A1 AROMATIC RING COMPOUND TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2013-08-29 WO disclosed