SCHEMBL28073642

SCHEMBL28073642

C=Cc1ccc2c(OC(=O)CCC)csc2c1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALOX15 P16050 2/20 0.40
LMNA P02545 1/20 0.38
ESR1 P03372 1/20 0.37
TOP2A P11388 3/20 0.36
TAS1R3 Q7RTX0 1/20 0.35
TAS1R1 Q7RTX1 1/20 0.35
TRPA1 O75762 1/20 0.34
ALDH1A1 P00352 2/20 0.34
KDM4E B2RXH2 2/20 0.34
KMT2A Q03164 2/20 0.34
GLA P06280 1/20 0.34
GAA P10253 1/20 0.34
AKR1C3 P42330 3/20 0.33
CA2 P00918 2/20 0.33
BCL9 O00512 1/20 0.33
CTNNB1 P35222 1/20 0.33
AKR1C2 P52895 1/20 0.33
MAPT P10636 1/20 0.33
HSD17B10 Q99714 1/20 0.33
VCP P55072 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31518877 0.80 ALOX15 (0.56) ALOX15TOP2ATRPA1ALDH1A1KDM4E
SCHEMBL28073631 0.78 CYP3A4 (0.40) ALOX15LMNAALDH1A1KDM4EKMT2A
SCHEMBL6990012 0.77 TOP2A (0.57) ALOX15TOP2ATRPA1KDM4EKMT2A
SCHEMBL9751544 0.74 ALOX15 (0.43) ALOX15LMNAALDH1A1KDM4EKMT2A
SCHEMBL28073641 0.74 PKM (0.39) ALOX15LMNAALDH1A1KDM4EKMT2A
SCHEMBL17431373 0.73 PTGS2 (0.33) TAS1R3TAS1R1ALDH1A1AKR1C3AKR1C2
SCHEMBL15211548 0.72 ESR1 (0.40) LMNAESR1ALDH1A1KDM4EKMT2A
SCHEMBL1703804 0.72 BCL9 (0.55) LMNAESR1TAS1R3TAS1R1ALDH1A1
SCHEMBL14732611 0.71 TDP1 (0.43) LMNAALDH1A1KDM4EKMT2AGLA
SCHEMBL27992465 0.71 KMT2A (0.40) ALOX15LMNAESR1ALDH1A1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104254525-B aromatic ring compound TAKEDA PHARMACEUTICAL CO.,LTD. (JP) 2016-05-25 CN disclosed