SCHEMBL15212089

SCHEMBL15212089

COc1c(Cl)cccc1S(=O)(=O)Nc1cccnc1

nearest known ligand 0.76

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.76
KMT2A Q03164 1/20 0.76
ALPL P05186 13/20 0.65
LMNA P02545 1/20 0.62
TP53 P04637 1/20 0.58
TDP1 Q9NUW8 1/20 0.58
GAA P10253 2/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL856880 0.86 ALDH1A1 (0.71) ALDH1A1KMT2AALPLLMNATP53
SCHEMBL1404359 0.77 ALPL (1.00) ALDH1A1ALPLLMNAGAA
SCHEMBL15211944 0.76 ALPL (1.00) ALDH1A1ALPLLMNAGAA
SCHEMBL15212055 0.76 ALPL (1.00) ALDH1A1ALPLLMNAGAA
SCHEMBL31371215 0.76 ALPL (1.00) ALDH1A1ALPLLMNAGAA
SCHEMBL15212153 0.76 ALPL (0.80) ALDH1A1KMT2AALPLLMNAGAA
SCHEMBL15212142 0.75 ALPL (0.66) ALPLLMNA
SCHEMBL3448568 0.74 ALDH1A1 (1.00) ALDH1A1KMT2AALPLLMNATP53
SCHEMBL31368924 0.74 ALDH1A1 (1.00) ALDH1A1KMT2AALPLLMNATP53
SCHEMBL15212110 0.73 ALPL (0.70) ALDH1A1KMT2AALPLLMNAGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 13 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-10370333-B2 Sulfonamide compounds and uses as TNAP inhibitors SANFORD-BURNHAM PREBYS MEDICAL DISCOVERY INSTITUTE (US) 2019-08-06 US disclosed
US-10370333-B2 Sulfonamide compounds and uses as TNAP inhibitors SANFORD-BURNHAM PREBYS MEDICAL DISCOVERY INSTITUTE (US) 2019-08-06 US disclosed
US-20190010126-A1 SULFONAMIDE COMPOUNDS AND USES AS TNAP INHIBITORS Sanford Burnham Prebys Medical Discovery Institute 2019-01-10 US disclosed
US-9884826-B2 Sulfonamide compounds and uses as TNAP inhibitors SANFORD-BURNHAM MEDICAL RESEARCH INSTITUTE (US) 2018-02-06 US disclosed
US-9884826-B2 Sulfonamide compounds and uses as TNAP inhibitors SANFORD-BURNHAM MEDICAL RESEARCH INSTITUTE (US) 2018-02-06 US disclosed
US-20160355479-A1 SULFONAMIDE COMPOUNDS AND USES AS TNAP INHIBITORS SANFORD-BURNHAM MEDICAL RESEARCH INSTITUTE 2016-12-08 US disclosed
US-20160355479-A1 SULFONAMIDE COMPOUNDS AND USES AS TNAP INHIBITORS SANFORD-BURNHAM MEDICAL RESEARCH INSTITUTE 2016-12-08 US disclosed
US-9458147-B2 Sulfonamide compounds and uses as TNAP inhibitors SANFORD-BURNHAM MEDICAL RESEARCH INSTITUTE (US) 2016-10-04 US disclosed
US-9458147-B2 Sulfonamide compounds and uses as TNAP inhibitors SANFORD-BURNHAM MEDICAL RESEARCH INSTITUTE (US) 2016-10-04 US disclosed
US-20150011551-A1 SULFONAMIDE COMPOUNDS AND USES AS TNAP INHIBITORS Sanford- Burnham Medical Reseach Institute (US) 2015-01-08 US disclosed
US-20150011551-A1 SULFONAMIDE COMPOUNDS AND USES AS TNAP INHIBITORS Sanford- Burnham Medical Reseach Institute (US) 2015-01-08 US disclosed
EP-2817292-A1 SULFONAMIDE COMPOUNDS AND USES AS TNAP INHIBITORS Sanford-Burnham Medical Research Institute (US) 2014-12-31 EP disclosed
WO-2013126608-A1 SULFONAMIDE COMPOUNDS AND USES AS TNAP INHIBITORS SANFORD-BURNHAM MEDICAL RESEARCH INSTITUTE (US) 2013-08-29 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-10370333-B2 Sulfonamide compounds and uses as TNAP inhibitors TNNI3, TNKS1BP1, TNNT2 ALDH1A1 3674/4885KMT2A 857/4885ALPL 503/4885
US-20150011551-A1 SULFONAMIDE COMPOUNDS AND USES AS TNAP INHIBITORS TNNI3, TNKS1BP1, TNNT2 ALDH1A1 3674/4885KMT2A 857/4885ALPL 503/4885
US-20190010126-A1 SULFONAMIDE COMPOUNDS AND USES AS TNAP INHIBITORS TNNI3, TNKS1BP1, TNNT2 ALDH1A1 3674/4885KMT2A 857/4885ALPL 503/4885
US-20160355479-A1 SULFONAMIDE COMPOUNDS AND USES AS TNAP INHIBITORS TNNI3, TNKS1BP1, TNNT2 ALDH1A1 3674/4885KMT2A 857/4885ALPL 503/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.