SCHEMBL15224176

SCHEMBL15224176

NCCCNC(=S)NCC1CCCCC1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 1/20 0.45
CA12 O43570 1/20 0.42
CA1 P00915 1/20 0.42
CA2 P00918 1/20 0.42
MMP1 P03956 1/20 0.42
MMP2 P08253 1/20 0.42
MMP3 P08254 1/20 0.42
MMP9 P14780 1/20 0.42
MMP8 P22894 1/20 0.42
CA9 Q16790 1/20 0.42
EPHX1 P07099 2/20 0.41
MEN1 O00255 2/20 0.40
KMT2A Q03164 2/20 0.40
SIGMAR1 Q99720 1/20 0.40
SMN1; SMN2 Q16637 2/20 0.40
ALDH1A1 P00352 2/20 0.40
MAPT P10636 2/20 0.40
HTT P42858 2/20 0.40
HPGD P15428 1/20 0.40
ALOX12 P18054 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7783075 0.83 CA12 (0.55) CYP2D6CA12CA1CA2MMP1
SCHEMBL6538230 0.80 CA12 (0.46) CYP2D6CA12CA1CA2MMP1
SCHEMBL6539544 0.80 CA12 (0.46) CYP2D6CA12CA1CA2MMP1
SCHEMBL7151996 0.78 CA12 (0.43) CYP2D6CA12CA1CA2MMP1
SCHEMBL10936950 0.77 SIGMAR1 (0.48) CYP2D6CA12CA1CA2CA9
SCHEMBL6974114 0.77 SIGMAR1 (0.48) CYP2D6CA12CA1CA2CA9
SCHEMBL15224187 0.77 KMT2A (0.67) MEN1KMT2ASMN1; SMN2ALDH1A1HTT
SCHEMBL15224173 0.77 CA2 (0.47) CYP2D6CA12CA1CA2MMP1
SCHEMBL18531459 0.76 ADAMTS4 (0.40) CA12CA1CA2MMP1MMP2
SCHEMBL21709912 0.76 ADAMTS4 (0.40) CA12CA1CA2MMP1MMP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2439202-B1 INHIBITOR COMPOUNDS OF 11-BETA-HYDROXYSTEROID DEHYDROGENASE TYPE 1 SALVAT LAB SA (ES) 2016-04-20 EP disclosed
US-8524894-B2 Inhibitor compounds of 11-beta-hydroxysteroid dehydrogenase type 1 LABORATORIOS SALVAT, S.A. (ES) 2013-09-03 US disclosed