SCHEMBL15225596

SCHEMBL15225596

CCc1c(O)cc(O)c(C(=O)c2ccc(OC)cc2)c1C(C)C(=O)O

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 2/20 0.41
CYP2C19 P33261 2/20 0.41
CYP3A4 P08684 1/20 0.41
PTGS2 P35354 5/20 0.40
PTGS1 P23219 4/20 0.40
AKR1C3 P42330 2/20 0.40
AKR1C2 P52895 2/20 0.40
HTT P42858 2/20 0.40
CYP1A2 P05177 2/20 0.40
GAA P10253 2/20 0.40
CDC42 P60953 1/20 0.40
RAC1 P63000 1/20 0.40
MAPT P10636 1/20 0.40
TSHR P16473 1/20 0.40
SLC22A6 Q4U2R8 1/20 0.40
SLC22A12 Q96S37 4/20 0.40
CNR2 P34972 1/20 0.39
ALDH1A1 P00352 2/20 0.39
LMNA P02545 1/20 0.39
PGR P06401 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15225780 0.87 STS (0.43) CYP2D6CYP2C19PTGS2PTGS1HTT
SCHEMBL15225813 0.86 PTGS2 (0.49) CYP2D6CYP2C19CYP3A4PTGS2PTGS1
SCHEMBL2861272 0.79 MAPT (0.47) CYP2D6CYP2C19CYP3A4AKR1C3AKR1C2
SCHEMBL2865471 0.75 CYP3A4 (0.45) CYP2D6CYP2C19CYP3A4AKR1C3AKR1C2
SCHEMBL2858867 0.75 NFKB1 (0.43) CYP2D6CYP2C19CYP3A4HTTGAA
SCHEMBL15225837 0.74 PTGS2 (0.51) CYP2D6CYP2C19CYP3A4PTGS2PTGS1
SCHEMBL2862959 0.73 PTGS2 (0.42) CYP2D6CYP2C19CYP3A4PTGS2HTT
SCHEMBL2858510 0.72 PTGS2 (0.43) CYP2D6CYP2C19CYP3A4PTGS2HTT
SCHEMBL2864661 0.71 LMNA (0.40) CYP2D6CYP2C19CYP3A4HTTGAA
SCHEMBL2868754 0.71 NFKB1 (0.40) CYP2D6CYP2C19CYP3A4HTTGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1642880-B1 HSP90 FAMILY PROTEIN INHIBITORS KYOWA HAKKO KIRIN CO LTD (JP) 2013-09-04 EP claimed