SCHEMBL15225813

SCHEMBL15225813

CCc1c(O)cc(O)c(C(=O)c2ccccc2)c1C(C)C(=O)O

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 6/20 0.49
PTGS1 P23219 5/20 0.49
SMN1; SMN2 Q16637 3/20 0.46
MAPT P10636 2/20 0.46
CXCR1 P25024 2/20 0.46
CXCR2 P25025 2/20 0.46
CYP3A4 P08684 2/20 0.46
HPGD P15428 2/20 0.46
ALDH1A1 P00352 2/20 0.46
RECQL P46063 1/20 0.46
KDM4E B2RXH2 1/20 0.46
LMNA P02545 1/20 0.46
MAPK1 P28482 1/20 0.46
PMP22 Q01453 1/20 0.46
SLC22A6 Q4U2R8 1/20 0.46
HSD17B10 Q99714 1/20 0.46
CXCL8 P10145 1/20 0.46
THPO P40225 1/20 0.46
HIF1A Q16665 1/20 0.46
ADRA2C P18825 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15225596 0.86 CYP2D6 (0.41) PTGS2PTGS1MAPTCYP3A4HPGD
SCHEMBL15225780 0.85 STS (0.43) PTGS2PTGS1SMN1; SMN2HPGDALDH1A1
SCHEMBL2862917 0.75 HPGD (0.40) PTGS2SMN1; SMN2MAPTCYP3A4HPGD
SCHEMBL2862066 0.71 LMNA (0.40) PTGS2SMN1; SMN2MAPTCYP3A4HPGD
SCHEMBL2863503 0.71 L3MBTL1 (0.40) SMN1; SMN2MAPTCYP3A4HPGDALDH1A1
SCHEMBL28132998 0.70 BCL2 (0.54) PTGS2PTGS1MAPTCYP3A4HPGD
SCHEMBL2862470 0.69 HPGD (0.49) PTGS2PTGS1SMN1; SMN2MAPTCYP3A4
SCHEMBL28001032 0.69 CES2 (0.44) HPGDALDH1A1KDM4EMAPK1HSD17B10
SCHEMBL2859684 0.69 GAA (0.40) PTGS2PTGS1SMN1; SMN2MAPTCYP3A4
SCHEMBL2857183 0.68 L3MBTL1 (0.37) SMN1; SMN2HPGDALDH1A1LMNAPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1642880-B1 HSP90 FAMILY PROTEIN INHIBITORS KYOWA HAKKO KIRIN CO LTD (JP) 2013-09-04 EP claimed