SCHEMBL15280356

SCHEMBL15280356

Cc1cnc(Cl)nc1OCCc1ccc(Oc2ccc(Cl)c(CF)c2)cc1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PLA2G7 Q13093 2/20 0.37
PIN1 Q13526 2/20 0.37
AXL P30530 1/20 0.34
PPARA Q07869 6/20 0.33
PPARG P37231 3/20 0.33
GPR84 Q9NQS5 2/20 0.33
POLB P06746 2/20 0.33
CASP6 P55212 1/20 0.33
RXRA P19793 1/20 0.32
GRIN1 Q05586 1/20 0.32
GRIN2B Q13224 1/20 0.32
NOS3 P29474 1/20 0.32
NOS1 P29475 1/20 0.32
FFAR1 O14842 1/20 0.31
KDM4E B2RXH2 1/20 0.31
PPARD Q03181 2/20 0.31
PDE2A O00408 1/20 0.31
HTR2A P28223 1/20 0.31
SLC6A4 P31645 1/20 0.31
KCNH2 Q12809 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9900476 0.84 PLA2G7 (0.51) PLA2G7PIN1GPR84
SCHEMBL9901043 0.74 KDM4E (0.37) PIN1AXLPPARAPPARGPOLB
SCHEMBL9905581 0.72 PLA2G7 (0.52) PLA2G7PIN1GPR84POLBCASP6
SCHEMBL15277225 0.71 GPR84 (0.43) PLA2G7PPARAPPARGGPR84POLB
SCHEMBL15278085 0.70 PLA2G7 (0.38) PLA2G7PPARAPPARGGPR84PPARD
SCHEMBL9900905 0.70 PIN1 (0.51) PIN1PPARGPOLBCASP6FFAR1
SCHEMBL15277253 0.69 GPR84 (0.42) PLA2G7PPARAPPARGGPR84POLB
SCHEMBL15278039 0.68 ST14 (0.55)
SCHEMBL15278102 0.68 PLA2G7 (0.57) PLA2G7PPARAPPARGGPR84
SCHEMBL9901204 0.67 POLB (0.45) PIN1POLBCASP6SLC6A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8859573-B2 Pyrimidinone and pyridinone compounds for use in the treatment of diseases or conditions mediated by Lp-PLA2 GLAXO GROUP LIMITED (GB) 2014-10-14 US disclosed
US-20130252986-A1 COMPOUNDS GLAXO GROUP LIMITED (GB) 2013-09-26 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20130252986-A1 COMPOUNDS LIPG, ENPP2, PLA2G1B PLA2G7 6/4885PIN1 1366/4885AXL 4424/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.