SCHEMBL15313898

SCHEMBL15313898

O=C(Nc1ccc2c(c1)S(=O)(=O)c1ccccc1-2)c1cc(-c2ccc3ccccc3c2)c(O)c(O)c1O

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAOA P21397 2/20 0.46
NPC1 O15118 7/20 0.45
RAB9A P51151 7/20 0.45
KMT2A Q03164 4/20 0.45
MEN1 O00255 3/20 0.45
PARG Q86W56 4/20 0.41
ALDH1A1 P00352 2/20 0.40
LMNA P02545 2/20 0.40
SMN1; SMN2 Q16637 2/20 0.40
KDM4E B2RXH2 1/20 0.40
GAA P10253 1/20 0.40
MAPT P10636 1/20 0.40
HDAC4 P56524 1/20 0.40
HDAC2 Q92769 1/20 0.40
HDAC8 Q9BY41 1/20 0.40
SLC6A2 P23975 1/20 0.39
SLC6A4 P31645 1/20 0.39
SLC6A3 Q01959 1/20 0.39
USP2 O75604 1/20 0.39
TP53 P04637 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15313875 0.84 MAOA (0.47) MAOANPC1RAB9AKMT2AMEN1
SCHEMBL15313899 0.75 BCL2 (0.67) MAOAKMT2AALDH1A1LMNASMN1; SMN2
SCHEMBL15313887 0.73 BCL2 (0.56) MAOANPC1KMT2AMEN1ALDH1A1
SCHEMBL13576567 0.72 MEN1 (0.63) MAOANPC1RAB9AKMT2AMEN1
SCHEMBL15313867 0.71 PARG (0.49) NPC1RAB9AKMT2AMEN1PARG
SCHEMBL15313854 0.70 BCL2L1 (0.64) NPC1RAB9AKMT2AMEN1PARG
SCHEMBL4869345 0.68 CA12 (0.68) MAOANPC1RAB9AKMT2AMEN1
SCHEMBL15313972 0.67 BCL2 (0.75) NPC1RAB9AKMT2AMEN1ALDH1A1
SCHEMBL7643064 0.66 NPC1 (0.81) NPC1RAB9AKMT2AMEN1ALDH1A1
SCHEMBL22911505 0.66 NPC1 (0.61) NPC1RAB9AKMT2AMEN1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8557812-B2 Small molecule inhibitors of anti-apoptotic BCL-2 family members and the uses thereof THE REGENTS OF THE UNIVERSITY OF MICHIGAN (US) 2013-10-15 US disclosed
US-8557812-B2 Small molecule inhibitors of anti-apoptotic BCL-2 family members and the uses thereof THE REGENTS OF THE UNIVERSITY OF MICHIGAN (US) 2013-10-15 US disclosed