SCHEMBL15314545

SCHEMBL15314545

CC(C)(CC(=O)NC1C2CC=C3CCC1C3C2)Cc1nc(-c2ccccn2)no1

nearest known ligand 0.68

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
HSD11B1 P28845 4/20 0.68
NPC1 O15118 9/20 0.44
RAB9A P51151 9/20 0.44
SMN1; SMN2 Q16637 7/20 0.44
HTT P42858 1/20 0.44
BMP1 P13497 1/20 0.37
ALDH1A1 P00352 3/20 0.37
EPHX2 P34913 3/20 0.35
HCRTR1 O43613 1/20 0.35
PRCP P42785 1/20 0.35
CYP3A4 P08684 1/20 0.34
KCNH2 Q12809 1/20 0.34
CACNA1C Q13936 1/20 0.34
KDM4E B2RXH2 1/20 0.34
TSHR P16473 1/20 0.34
TP53 P04637 1/20 0.34
MAPK1 P28482 1/20 0.34
GAA P10253 1/20 0.34
POLB P06746 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14159668 0.82 HSD11B1 (0.79) HSD11B1NPC1RAB9ASMN1; SMN2HTT
SCHEMBL3616180 0.81 HSD11B1 (1.00) HSD11B1NPC1RAB9ASMN1; SMN2HTT
SCHEMBL3623669 0.64 HSD11B1 (0.84) HSD11B1HTTALDH1A1TSHR
SCHEMBL3621674 0.64 HSD11B1 (0.73) HSD11B1SMN1; SMN2HTTTSHRMAPK1
SCHEMBL3620712 0.63 HSD11B1 (0.64) HSD11B1NPC1RAB9ASMN1; SMN2BMP1
SCHEMBL3612338 0.60 HSD11B1 (1.00) HSD11B1EPHX2
SCHEMBL6313243 0.60 HPGD (0.59) NPC1RAB9ASMN1; SMN2HTTALDH1A1
SCHEMBL3518102 0.60 HSD11B1 (0.49) HSD11B1NPC1RAB9ASMN1; SMN2HTT
SCHEMBL4034138 0.60 NPC1 (0.65) NPC1RAB9ASMN1; SMN2HTTALDH1A1
SCHEMBL29463848 0.59 RAB9A (1.00) NPC1RAB9ASMN1; SMN2HTTBMP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2094263-B1 2-ADAMANTYL-BUTYRAMIDE DERIVATIVES AS SELECTIVE 11 BETA-HSD1 INHIBITORS MERCK PATENT GMBH (DE) 2013-10-16 EP disclosed