SCHEMBL15410033

SCHEMBL15410033

O=C(Nc1c(F)c(F)c(C(F)(F)F)c(F)c1F)c1ccccc1

nearest known ligand 0.54

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 5/20 0.54
RAB9A P51151 5/20 0.54
P2RX1 P51575 1/20 0.51
TSHR P16473 1/20 0.48
NPSR1 Q6W5P4 1/20 0.48
KCNJ11 Q14654 1/20 0.47
KCNK3 O14649 3/20 0.47
LMNA P02545 3/20 0.46
KMT2A Q03164 2/20 0.46
MEN1 O00255 1/20 0.46
MAPT P10636 1/20 0.46
HPGD P15428 1/20 0.45
MDM4 O15151 1/20 0.45
TP53 P04637 1/20 0.45
KCNK9 Q9NPC2 2/20 0.44
HDAC1 Q13547 1/20 0.44
HDAC8 Q9BY41 1/20 0.44
HDAC6 Q9UBN7 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4586310 0.86 TSHR (0.60) NPC1RAB9ATSHRNPSR1KCNK3
SCHEMBL15410493 0.84 TSHR (0.42) NPC1RAB9ATSHRNPSR1LMNA
SCHEMBL15409614 0.84 RAB9A (0.52) NPC1RAB9AKCNJ11LMNAKMT2A
SCHEMBL15410034 0.84 KCNJ11 (0.47) NPC1RAB9ANPSR1KCNJ11LMNA
SCHEMBL15410726 0.83 TRPV1 (0.59) NPC1RAB9ANPSR1KMT2AMEN1
SCHEMBL15411914 0.82 NPSR1 (0.55) NPC1RAB9AP2RX1TSHRNPSR1
SCHEMBL15411037 0.82 ABCC9 (0.52) RAB9ATSHRNPSR1KCNJ11KCNK3
SCHEMBL15410723 0.82 KCNJ11 (0.52) NPC1RAB9AP2RX1TSHRNPSR1
SCHEMBL15411277 0.82 KCNK3 (0.56) NPC1RAB9ATSHRNPSR1KCNJ11
SCHEMBL15412057 0.82 NPC1 (0.61) NPC1RAB9ALMNAKMT2AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20140018566-A1 PALLADIUM(II)-CATALYZED SELECTIVE FLUORINATION OF BENZOIC ACIDS AND DERIVATIVES THE SCRIPPS RESEARCH INSTITUTE (US) 2014-01-16 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20140018566-A1 PALLADIUM(II)-CATALYZED SELECTIVE FLUORINATION OF BENZOIC ACIDS AND DERIVATIVES AHR, DDT, AOC2 NPC1 2304/4885RAB9A 661/4885P2RX1 2449/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.