SCHEMBL15427985

SCHEMBL15427985

CNC(=O)c1[nH]c2ccc(O)cc2c1CCN

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR6 P50406 4/20 0.60
HTR1D P28221 3/20 0.60
HSD17B10 Q99714 3/20 0.60
CYP1A2 P05177 2/20 0.60
CYP3A4 P08684 2/20 0.60
CYP2D6 P10635 2/20 0.60
CYP2C9 P11712 2/20 0.60
HTR7 P34969 2/20 0.60
HTR3A P46098 2/20 0.60
TDP1 Q9NUW8 2/20 0.60
MAPK1 P28482 1/20 0.60
CYP2C19 P33261 1/20 0.60
NPSR1 Q6W5P4 3/20 0.57
RAD52 P43351 1/20 0.57
BLM P54132 1/20 0.57
SPR P35270 1/20 0.43
HTR1A P08908 2/20 0.43
HTR2A P28223 2/20 0.43
HTR2C P28335 2/20 0.43
HTR2B P41595 2/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16923032 0.87 EGFR (0.52) HTR6HTR1DHSD17B10CYP1A2CYP3A4
SCHEMBL16716149 0.84 HTR1D (0.61) HTR6HTR1DHSD17B10CYP1A2CYP3A4
SCHEMBL4292563 0.83 HTR6 (0.62) HTR6HTR1DHSD17B10CYP1A2CYP3A4
Hydrochloric Acid SCHEMBL16711692 0.83 HTR1D (0.60) HTR6HTR1DHSD17B10CYP1A2CYP3A4
SCHEMBL16711712 0.80 SPR (0.47) HSD17B10CYP1A2CYP3A4CYP2D6NPSR1
SCHEMBL18235616 0.80 TRPM8 (0.66) HTR6HSD17B10CYP1A2CYP2C9NPSR1
Hydrochloric Acid SCHEMBL18222557 0.79 TRPM8 (0.65) HTR6HSD17B10CYP1A2CYP2C9NPSR1
SCHEMBL16923054 0.78 HTR6 (0.41) HTR6HTR1DHSD17B10CYP1A2CYP3A4
SCHEMBL29361176 0.76 HTR6 (1.00) HTR6HTR1DHSD17B10CYP1A2CYP3A4
SCHEMBL399028 0.76 HTR6 (1.00) HTR6HTR1DHSD17B10CYP1A2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2014010602-A1 INDOLECARBOXAMIDE DERIVATIVE アステラス製薬株式会社 (JP) 2014-01-16 WO disclosed