SCHEMBL1551591

SCHEMBL1551591

Cc1nc2ccccc2c(=O)n1-c1ccccc1Br

nearest known ligand 0.73

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.73
L3MBTL1 Q9Y468 3/20 0.73
LMNA P02545 2/20 0.73
TSHR P16473 1/20 0.60
GLA P06280 1/20 0.59
HCAR1 Q9BXC0 1/20 0.57
MEN1 O00255 1/20 0.56
KMT2A Q03164 1/20 0.56
POLB P06746 1/20 0.56
PDE7A Q13946 1/20 0.55
HSD17B10 Q99714 1/20 0.55
MAPK1 P28482 1/20 0.55
ALOX12 P18054 1/20 0.55
NPSR1 Q6W5P4 1/20 0.55
HPD P32754 1/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30726101 1.00 ALDH1A1 (0.73) ALDH1A1L3MBTL1LMNATSHRGLA
SCHEMBL123247 0.90 ALDH1A1 (0.68) ALDH1A1L3MBTL1LMNATSHRGLA
Methaqualone SCHEMBL43892 0.84 ALDH1A1 (1.00) ALDH1A1L3MBTL1LMNATSHRGLA
Methaqualone SCHEMBL29386732 0.84 ALDH1A1 (1.00) ALDH1A1L3MBTL1LMNATSHRGLA
Methaqualone SCHEMBL20471677 0.84 ALDH1A1 (1.00) ALDH1A1L3MBTL1LMNATSHRGLA
Methaqualone SCHEMBL29355239 0.84 ALDH1A1 (1.00) ALDH1A1L3MBTL1LMNATSHRGLA
SCHEMBL6601150 0.84 L3MBTL1 (0.62) ALDH1A1L3MBTL1LMNAGLAHCAR1
SCHEMBL16596956 0.83 L3MBTL1 (0.77) ALDH1A1L3MBTL1LMNATSHRGLA
Methaqualone SCHEMBL3500629 0.83 ALDH1A1 (0.97) ALDH1A1L3MBTL1LMNATSHRGLA
Methaqualone SCHEMBL29849847 0.83 ALDH1A1 (0.97) ALDH1A1L3MBTL1LMNATSHRGLA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 91 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020006606-A1 A PHARMACEUTICAL COMPOSITION AND METHOD OF USE OF SAME HELIUM 3 RESOURCES PTY LTD (AU) 2020-01-09 WO claimed
US-20120095104-A1 USE OF VASOCONSTRICTORS ZACHAR ORON (IL) 2012-04-19 US claimed
EP-2376073-A2 DERMAL APPLICATION OF VASOCONSTRICTORS Zachar, Oron (IL) 2011-10-19 EP claimed
US-20110144209-A1 USE OF VASOCONSTRICTORS ZACHAR ORON 2011-06-16 US claimed
EP-2313037-A1 DERMAL APPLICATION OF VASOCONSTRICTORS Zachar, Oron (IL) 2011-04-27 EP claimed
WO-2010063030-A2 DERMAL APPLICATION OF VASOCONSTRICTORS FEIGELSON, DANIEL (IL) 2010-06-03 WO claimed
WO-2010001391-A1 DERMAL APPLICATION OF VASOCONSTRICTORS ZACHAR ORON (IL) 2010-01-07 WO claimed
US-20250367232-A1 HALOGEN TREATMENT OF HEART ATTACK AND ISCHEMIC INJURY HUTCHINSON FRED CANCER RES (US) 2025-12-04 US disclosed
US-20250255928-A1 USE OF COLLAGEN HYDROLYSATE AS AN ACTIVE INGREDIENT IN AMELIORATING SLEEP ROUSSELOT B.V. (BE) 2025-08-14 US disclosed
US-12377235-B2 Multipurpose device INSTITUTE FOR CANCER RESEARCH (US) 2025-08-05 US disclosed
EP-4463177-B1 USE OF COLLAGEN HYDROLYSATE AS AN ACTIVE INGREDIENT IN AMELIORATING SLEEP ROUSSELOT BV (BE) 2025-05-14 EP disclosed
US-20250032419-A1 SOLID PHARMACEUTICAL COMPOSITIONS AND METHODS OF PRODUCING THE SAME GALVITA AG (CH) 2025-01-30 US disclosed
EP-4463177-A1 USE OF COLLAGEN HYDROLYSATE AS AN ACTIVE INGREDIENT IN AMELIORATING SLEEP Rousselot BV (BE) 2024-11-20 EP disclosed
US-20120095104-A1 USE OF VASOCONSTRICTORS ZACHAR ORON (IL) 2012-04-19 US disclosed
CN-102300566-A Cutaneous application of vasoconstrictors 2011-12-28 CN disclosed
EP-2376073-A2 DERMAL APPLICATION OF VASOCONSTRICTORS Zachar, Oron (IL) 2011-10-19 EP disclosed
US-20110144209-A1 USE OF VASOCONSTRICTORS ZACHAR ORON 2011-06-16 US disclosed
EP-2313037-A1 DERMAL APPLICATION OF VASOCONSTRICTORS Zachar, Oron (IL) 2011-04-27 EP disclosed
WO-2010063030-A2 DERMAL APPLICATION OF VASOCONSTRICTORS FEIGELSON, DANIEL (IL) 2010-06-03 WO disclosed
WO-2010001391-A1 DERMAL APPLICATION OF VASOCONSTRICTORS ZACHAR ORON (IL) 2010-01-07 WO disclosed