Pentobarbital

Pentobarbital

SCHEMBL15533339

CC(=O)c1ccccc1.CCCC(C)C1(CC)C(=O)N=C([O-])NC1=O.[Na+]

nearest known ligand 0.46

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

GABRA1GABRA2GABRA3GABRA4GABRA5GABRA6GABRB1GABRB2GABRB3GABRDGABREGABRG1GABRG2GABRG3GABRPGABRQ

The experimentally established mechanism targets of Pentobarbital. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GABRB3 known ✓ P28472 1/20 0.42
GABRA2 known ✓ P47869 1/20 0.42
GABRB2 known ✓ P47870 1/20 0.42
LMNA P02545 5/20 0.46
CYP3A4 P08684 3/20 0.42
KDM4E B2RXH2 1/20 0.42
ALDH1A1 P00352 1/20 0.42
OPRD1 P41143 1/20 0.42
RECQL P46063 1/20 0.40
MMP9 P14780 1/20 0.33
KMT2A Q03164 3/20 0.32
GLA P06280 1/20 0.32
THRB P10828 1/20 0.32
CYP2C9 P11712 1/20 0.32
BLM P54132 1/20 0.32
PMP22 Q01453 1/20 0.32
NR1I2 O75469 1/20 0.31
POLB P06746 1/20 0.31
PKM P14618 1/20 0.31
MEN1 O00255 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Pentobarbital SCHEMBL8081141 0.92 LMNA (0.47) LMNACYP3A4KDM4EALDH1A1GABRB3
Pentobarbital SCHEMBL477033 0.89 CYP3A4 (0.50) LMNACYP3A4KDM4EALDH1A1GABRB3
Pentobarbital SCHEMBL1451667 0.89 CYP3A4 (0.53) LMNACYP3A4KDM4EALDH1A1GABRB3
Pentobarbital SCHEMBL7152508 0.88 CYP3A4 (0.45) LMNACYP3A4KDM4EALDH1A1GABRB3
Pentobarbital SCHEMBL1836479 0.88 LMNA (0.49) LMNACYP3A4KDM4EALDH1A1GABRB3
Pentobarbital SCHEMBL2769858 0.87 CYP3A4 (0.51) LMNACYP3A4KDM4EALDH1A1GABRB3
Pentobarbital SCHEMBL10727223 0.87 CYP3A4 (0.51) LMNACYP3A4KDM4EALDH1A1GABRB3
Pentobarbital SCHEMBL4202506 0.86 LMNA (0.44) LMNACYP3A4KDM4EALDH1A1GABRB3
Pentobarbital SCHEMBL2126265 0.86 LMNA (0.49) LMNACYP3A4KDM4EALDH1A1GABRB3
Pentobarbital SCHEMBL2689394 0.85 CYP3A4 (0.49) LMNACYP3A4KDM4EALDH1A1GABRB3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9725383-B2 Oxygenates-free C8-C12 aromatic hydrocarbon stream and a process for preparing the same RELIANCE INDUSTRIES LIMITED (IN) 2017-08-08 US disclosed
US-20150073197-A1 Oxygenates-Free C8-C12 Aromatic Hydrocarbon Stream and a Process for Preparing the Same RELIANCE INDUSTRIES LIMITED (IN) 2015-03-12 US disclosed
EP-2834211-A1 AN OXYGENATES-FREE C8-C12 AROMATIC HYDROCARBON STREAM AND A PROCESS FOR PREPARING THE SAME Reliance Industries Limited (IN) 2015-02-11 EP disclosed
WO-2013175490-A1 AN OXYGENATES-FREE C8-C12 AROMATIC HYDROCARBON STREAM AND A PROCESS FOR PREPARING THE SAME RELIANCE INDUSTRIES LIMITED (IN) 2013-11-28 WO disclosed