SCHEMBL15533871

SCHEMBL15533871

FC(F)(F)c1cccc(Nc2cc(-c3ccccc3)ncn2)n1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TP53 P04637 3/20 0.51
MAPT P10636 2/20 0.51
ABL1 P00519 6/20 0.49
BCR P11274 6/20 0.49
JAK2 O60674 1/20 0.47
TAS2R14 Q9NYV8 1/20 0.47
TRPV1 Q8NER1 2/20 0.46
FAAH O00519 2/20 0.44
USP2 O75604 2/20 0.43
CYP2D6 P10635 2/20 0.43
CYP2C19 P33261 2/20 0.43
CYP1A2 P05177 1/20 0.43
CYP3A4 P08684 1/20 0.43
CYP2C9 P11712 1/20 0.43
TSHR P16473 1/20 0.43
CLK4 Q9HAZ1 1/20 0.43
SYK P43405 2/20 0.43
ASIC3 Q9UHC3 1/20 0.43
MEN1 O00255 1/20 0.42
ALDH1A1 P00352 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15534259 0.90 TRPV1 (0.57) ABL1BCRTRPV1FAAH
SCHEMBL15534464 0.88 ABL1 (0.46) TP53MAPTABL1BCRJAK2
SCHEMBL15534267 0.88 TRPV1 (0.56) TP53MAPTABL1BCRJAK2
SCHEMBL15533815 0.86 TRPV1 (0.48) TP53MAPTABL1BCRJAK2
SCHEMBL15533746 0.85 SYK (0.48) MAPTABL1BCRTRPV1FAAH
SCHEMBL15533972 0.85 ABL1 (0.53) TP53MAPTABL1BCRFAAH
SCHEMBL15534101 0.85 TRPV1 (0.47) TP53MAPTABL1BCRJAK2
Bromide SCHEMBL15534396 0.84 TRPV1 (0.47) TP53MAPTABL1BCRJAK2
Hydrochloric Acid SCHEMBL15533549 0.84 TRPV1 (0.47) TP53MAPTABL1BCRJAK2
SCHEMBL15533969 0.83 CYP1A1 (0.48) TP53ABL1BCRFAAHCYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013175415-A1 SUBSTITUTED PYRIMIDINE COMPOUNDS AND USES THEREOF Piramal Enterprises Limited (IN) 2013-11-28 WO claimed
WO-2013175415-A1 SUBSTITUTED PYRIMIDINE COMPOUNDS AND USES THEREOF Piramal Enterprises Limited (IN) 2013-11-28 WO disclosed