SCHEMBL15533969

SCHEMBL15533969

COc1cc(OC)cc(-c2cc(Nc3cccc(C(F)(F)F)n3)ncn2)c1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A1 P04798 1/20 0.48
CYP1B1 Q16678 1/20 0.48
ABL1 P00519 8/20 0.44
BCR P11274 7/20 0.44
SYK P43405 3/20 0.44
CLK4 Q9HAZ1 5/20 0.43
CYP1A2 P05177 5/20 0.43
CYP3A4 P08684 5/20 0.43
CYP2D6 P10635 5/20 0.43
TSHR P16473 5/20 0.43
CYP2C19 P33261 5/20 0.43
MAPK1 P28482 3/20 0.43
TP53 P04637 2/20 0.43
HIF1A Q16665 1/20 0.43
HSD17B10 Q99714 1/20 0.43
LMNA P02545 2/20 0.42
GRM5 P41594 1/20 0.41
ALDH1A1 P00352 2/20 0.41
PLK4 O00444 1/20 0.41
DYRK3 O43781 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15533972 0.91 ABL1 (0.53) ABL1BCRSYKTP53SMN1; SMN2
SCHEMBL15533691 0.84 MAPT (0.47) ABL1BCRCLK4CYP1A2CYP3A4
SCHEMBL15533871 0.83 TP53 (0.51) ABL1BCRSYKCLK4CYP1A2
SCHEMBL15533818 0.82 CYP2D6 (0.50) SYKCLK4CYP1A2CYP3A4CYP2D6
SCHEMBL15533815 0.82 TRPV1 (0.48) ABL1BCRSYKMAPK1TP53
SCHEMBL15534259 0.81 TRPV1 (0.57) ABL1BCRFAAH
SCHEMBL15534453 0.80 TAS2R14 (0.47) ABL1BCRSYKTP53LMNA
SCHEMBL15534267 0.80 TRPV1 (0.56) ABL1BCRSYKTP53FAAH
SCHEMBL15534464 0.80 ABL1 (0.46) ABL1BCRSYKTP53
SCHEMBL15534101 0.79 TRPV1 (0.47) ABL1BCRMAPK1TP53FAAH

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013175415-A1 SUBSTITUTED PYRIMIDINE COMPOUNDS AND USES THEREOF Piramal Enterprises Limited (IN) 2013-11-28 WO claimed
WO-2013175415-A1 SUBSTITUTED PYRIMIDINE COMPOUNDS AND USES THEREOF Piramal Enterprises Limited (IN) 2013-11-28 WO disclosed