SCHEMBL1554487

SCHEMBL1554487

CC(C)Nc1nccc(C(C=O)=C(c2ccc(F)cc2)N(C)C)n1

nearest known ligand 0.37

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
MAPK14 Q16539 9/20 0.37
KCNH3 Q9ULD8 2/20 0.35
USP2 O75604 1/20 0.34
CYP1A2 P05177 1/20 0.34
CYP3A4 P08684 1/20 0.34
CYP2C19 P33261 1/20 0.34
GRM5 P41594 1/20 0.34
GRM1 Q13255 1/20 0.34
IDH1 O75874 4/20 0.32
HRH4 Q9H3N8 1/20 0.32
MAPK13 O15264 2/20 0.32
MAPK12 P53778 2/20 0.32
MAPK11 Q15759 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL709768 0.76 CES1 (0.43) MAPK14KCNH3IDH1HRH4
SCHEMBL1554486 0.76 MAPK14 (0.36) MAPK14KCNH3USP2CYP1A2CYP3A4
SCHEMBL1555485 0.76 MAPK14 (0.36) MAPK14KCNH3USP2CYP1A2CYP3A4
SCHEMBL5788690 0.70 LTA4H (0.49) USP2CYP1A2CYP2C19GRM1
SCHEMBL1554350 0.67 RAB9A (0.50) MAPK14KCNH3IDH1
SCHEMBL28748558 0.66 TRPV1 (0.33) MAPK14USP2CYP1A2CYP3A4CYP2C19
SCHEMBL27516993 0.66 TRPV1 (0.33) MAPK14USP2CYP1A2CYP3A4CYP2C19
SCHEMBL1554351 0.65 IDH1 (0.43) MAPK14KCNH3IDH1HRH4MAPK13
SCHEMBL8094065 0.64 LMNA (0.40) CYP1A2CYP2C19
SCHEMBL8094061 0.64 LMNA (0.40) CYP1A2CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2486031-A2 Phenylpyri(mi)dinylpyrazoles and their use as fungicides Bayer CropScience AG (DE) 2012-08-15 EP disclosed
WO-2011042389-A2 PHENYLPYRI(MI)DINYLAZOLES BAYER CROPSCIENCE AG (DE) 2011-04-14 WO disclosed