SCHEMBL15564679

SCHEMBL15564679

CCCCOC(=O)NC(CC(=O)O)Sc1c(N)cccc1N

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.43
HSD17B10 Q99714 2/20 0.43
CTSK P43235 2/20 0.40
RAB9A P51151 7/20 0.39
HPGD P15428 3/20 0.39
LMNA P02545 3/20 0.39
POLB P06746 2/20 0.39
KDM4E B2RXH2 1/20 0.39
SMN1; SMN2 Q16637 7/20 0.39
NPC1 O15118 6/20 0.39
L3MBTL1 Q9Y468 2/20 0.38
MAPK1 P28482 1/20 0.38
CYP1A2 P05177 3/20 0.37
CYP2C19 P33261 3/20 0.37
CYP2C9 P11712 2/20 0.37
TDP1 Q9NUW8 2/20 0.37
TSHR P16473 2/20 0.36
CYP3A4 P08684 1/20 0.36
PDE4D Q08499 1/20 0.36
MMEL1 Q495T6 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6654292 0.79 FAAH (0.42) CTSKRAB9AHPGDLMNAPOLB
SCHEMBL6654077 0.78 PLA2G10 (0.46) CTSKRAB9AHPGDLMNASMN1; SMN2
SCHEMBL7447309 0.77 CTSK (0.45) ALDH1A1HSD17B10CTSKRAB9AHPGD
SCHEMBL15564677 0.77 ALDH1A1 (0.43) ALDH1A1HSD17B10CTSKRAB9AHPGD
SCHEMBL6692027 0.76 EPHX1 (0.41) ALDH1A1CTSKRAB9AHPGDSMN1; SMN2
SCHEMBL2910068 0.71 CYP2C19 (0.47) ALDH1A1CTSKHPGDPOLBKDM4E
SCHEMBL844472 0.71 SMN1; SMN2 (0.57) ALDH1A1CTSKRAB9AHPGDLMNA
SCHEMBL14040614 0.71 SMN1; SMN2 (0.57) ALDH1A1CTSKRAB9AHPGDLMNA
SCHEMBL4265545 0.71 SMN1; SMN2 (0.50) ALDH1A1RAB9AHPGDLMNASMN1; SMN2
SCHEMBL6656147 0.71 FAAH (0.41) ALDH1A1HSD17B10CTSKRAB9AHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2882725-A1 SUBSTITUTED HETERO-AZEPINONES F. Hoffmann-La Roche AG (CH) 2015-06-17 EP disclosed
WO-2014023708-A1 SUBSTITUTED HETERO-AZEPINONES F. HOFFMANN-LA ROCHE AG (CH) 2014-02-13 WO disclosed