SCHEMBL15567698

SCHEMBL15567698

NC(=O)c1c(C(=O)O)cccc1-c1ccncc1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IKBKB O14920 3/20 0.48
CHUK O15111 3/20 0.48
IKBKE Q14164 1/20 0.48
PKMYT1 Q99640 1/20 0.48
BCAT2 O15382 1/20 0.47
HNF4A P41235 1/20 0.45
CCNC P24863 4/20 0.44
CDK8 P49336 4/20 0.44
ALDH1A1 P00352 2/20 0.44
PLK4 O00444 1/20 0.43
MAPK13 O15264 1/20 0.43
DYRK3 O43781 1/20 0.43
ROCK2 O75116 1/20 0.43
RPS6KA5 O75582 1/20 0.43
PRKD3 O94806 1/20 0.43
MAP4K4 O95819 1/20 0.43
CHEK2 O96017 1/20 0.43
PIM1 P11309 1/20 0.43
PHKG2 P15735 1/20 0.43
PRKACA P17612 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL570758 0.86 BCAT2 (0.63) BCAT2HNF4AALDH1A1SRCPARP1
SCHEMBL29916354 0.86 BCAT2 (0.63) BCAT2HNF4AALDH1A1SRCPARP1
SCHEMBL867477 0.81 MYC (0.47) BCAT2HNF4AALDH1A1PARP1MYC
SCHEMBL28115051 0.80 IKBKB (0.54) IKBKBCHUKIKBKEPKMYT1BCAT2
SCHEMBL15903687 0.80 CCNC (0.50) BCAT2CCNCCDK8ALDH1A1PIM1
Ethylamine SCHEMBL29028660 0.79 BCAT2 (0.54) BCAT2HNF4AALDH1A1MYCSMN1; SMN2
SCHEMBL6794827 0.79 ALDH1A1 (0.60) IKBKBCHUKIKBKEPKMYT1BCAT2
SCHEMBL8109600 0.78 HNF4A (0.49) IKBKBCHUKIKBKEPKMYT1HNF4A
SCHEMBL901580 0.78 BCAT2 (0.71) IKBKBCHUKIKBKEPKMYT1BCAT2
SCHEMBL164881 0.78 BCAT2 (0.71) IKBKBCHUKIKBKEPKMYT1BCAT2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2014025651-A1 CHROMAN DERIVATIVES AS TRPM8 INHIBITORS AMGEN INC. (US) 2014-02-13 WO disclosed