SCHEMBL15568264

SCHEMBL15568264

c1ccc(Cn2c(COc3cccc(-c4nc5ccccc5n4Cc4ccccc4)c3)nc3ccccc32)cc1

nearest known ligand 0.72

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
TP53 P04637 11/20 0.72
MAPT P10636 8/20 0.72
ALDH1A1 P00352 3/20 0.62
PDE6D O43924 1/20 0.62
ALDH2 P05091 1/20 0.62
ALDH3A1 P30838 1/20 0.62
GAA P10253 1/20 0.60
NPSR1 Q6W5P4 2/20 0.56
HPGD P15428 1/20 0.56
HTT P42858 1/20 0.56
SMN1; SMN2 Q16637 1/20 0.56
MEN1 O00255 1/20 0.53
KMT2A Q03164 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15568058 0.83 TP53 (0.63) TP53MAPTALDH1A1PDE6DALDH2
SCHEMBL15568494 0.82 TP53 (0.59) TP53MAPTALDH1A1PDE6DALDH2
SCHEMBL15568359 0.79 TP53 (0.76) TP53MAPTALDH1A1PDE6DALDH2
SCHEMBL15063430 0.79 TP53 (0.87) TP53MAPTSMN1; SMN2
SCHEMBL29412044 0.79 TP53 (1.00) TP53MAPTALDH1A1PDE6DALDH2
SCHEMBL28227635 0.79 TP53 (0.69) TP53MAPTALDH1A1PDE6DALDH2
SCHEMBL229828 0.78 ALDH1A1 (1.00) TP53MAPTALDH1A1PDE6DALDH2
SCHEMBL29412062 0.78 TP53 (0.78) TP53MAPTALDH1A1PDE6DALDH2
SCHEMBL15568102 0.77 TP53 (0.76) TP53MAPTALDH1A1PDE6DALDH2
SCHEMBL15673535 0.76 LMNA (0.72) TP53MAPTALDH1A1PDE6DALDH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2014027053-A1 BENZIMIDAZOLES FOR THE TREATMENT OF CANCER MAX-PLANCK-Gesellschaft zur Förderung der Wissenschaften e.V. (DE) 2014-02-20 WO claimed
WO-2014027053-A1 BENZIMIDAZOLES FOR THE TREATMENT OF CANCER MAX-PLANCK-Gesellschaft zur Förderung der Wissenschaften e.V. (DE) 2014-02-20 WO disclosed