SCHEMBL15580692

SCHEMBL15580692

CCc1ccc(-c2ccc(F)c(C(=O)O)c2)cc1Cl

nearest known ligand 0.47

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
SCN9A Q15858 1/20 0.47
SLC1A3 P43003 1/20 0.44
SLC1A2 P43004 1/20 0.44
SLC1A1 P43005 1/20 0.44
AKR1C2 P52895 5/20 0.43
AKR1C1 Q04828 5/20 0.43
MRGPRX4 Q96LA9 1/20 0.43
LMNA P02545 1/20 0.42
RARB P10826 2/20 0.42
RARA P10276 1/20 0.42
RARG P13631 1/20 0.42
RPA1 P27694 1/20 0.41
PDE4B Q07343 1/20 0.41
DCLRE1B Q9H816 1/20 0.40
FABP4 P15090 1/20 0.40
FABP5 Q01469 1/20 0.40
MCL1 Q07820 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11693510 0.80 AKR1C2 (0.52) SLC1A3SLC1A2SLC1A1AKR1C2AKR1C1
SCHEMBL2771168 0.76 KDM4E (0.52) DCLRE1BMCL1
SCHEMBL12603776 0.75 SCN9A (0.42) SCN9ASLC1A3SLC1A2SLC1A1
SCHEMBL12603775 0.75 AHR (0.50) SCN9ALMNA
SCHEMBL14072811 0.74 LMNA (0.43) LMNARARBRARARARGMCL1
SCHEMBL458111 0.73 ESR2 (0.52) AKR1C2AKR1C1DCLRE1B
SCHEMBL3062072 0.73 BCL2L1 (0.55) AKR1C2AKR1C1LMNAFABP4MCL1
SCHEMBL121427 0.73 ACMSD (0.63) AKR1C2AKR1C1DCLRE1BMCL1
SCHEMBL31028186 0.73 ACMSD (0.63) AKR1C2AKR1C1DCLRE1BMCL1
SCHEMBL5419835 0.73 FABP4 (0.47) AKR1C2AKR1C1MRGPRX4FABP4FABP5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2411365-B1 2,3-DIARYL- OR HETEROARYL-SUBSTITUTED 1,1,1-TRIFLUORO-2-HYDROXYPROPYL COMPOUNDS HOFFMANN LA ROCHE (CH) 2014-03-19 EP disclosed