SCHEMBL15635948

SCHEMBL15635948

NC(=O)c1cnc(NCCC(F)(F)F)nc1

nearest known ligand 0.45

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
ACACB O00763 2/20 0.45
VNN1 O95497 13/20 0.43
HDAC3 O15379 3/20 0.40
HDAC1 Q13547 3/20 0.40
HDAC2 Q92769 3/20 0.40
HDAC6 Q9UBN7 3/20 0.40
NNMT P40261 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL840255 0.85 ACACB (0.46) ACACBVNN1HDAC3HDAC1HDAC2
SCHEMBL13737548 0.74 HCAR3 (0.52) VNN1HDAC3HDAC1HDAC2
SCHEMBL13160092 0.74 VNN1 (0.48) ACACBVNN1HDAC3HDAC1HDAC2
SCHEMBL840192 0.74 ACACB (0.41) ACACBHDAC3HDAC1HDAC2HDAC6
SCHEMBL27770902 0.72 JAK3 (0.47) VNN1HDAC3HDAC1HDAC2HDAC6
SCHEMBL3668875 0.72 SCN9A (0.47) HDAC6NNMT
SCHEMBL2564257 0.71 ALDH1A1 (0.62) ACACBHDAC1HDAC6
SCHEMBL738119 0.71 STAT6 (0.57) VNN1HDAC3HDAC1HDAC2HDAC6
SCHEMBL30969276 0.71 CCNA2 (0.51) VNN1HDAC6
SCHEMBL4650847 0.70 NNMT (0.41) VNN1NNMT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2903965-A1 N-PROP-2-YNYL CARBOXAMIDE DERIVATIVES AND THEIR USE AS TRPA1 ANTAGONISTS Orion Corporation (FI) 2015-08-12 EP disclosed
WO-2014053694-A1 N-PROP-2-YNYL CARBOXAMIDE DERIVATIVES AND THEIR USE AS TRPA1 ANTAGONISTS ORION CORPORATION (FI) 2014-04-10 WO disclosed