SCHEMBL15740404

SCHEMBL15740404

O=CC(OC1CCC(Nc2ccc([N+](=O)[O-])c(C(F)(F)F)c2)CC1)N1CCN(CCc2nc3cc(C(F)(F)F)ccc3s2)CC1

nearest known ligand 0.36

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
TMEM97 Q5BJF2 8/20 0.36
CYP2C19 P33261 2/20 0.33
CYP1A2 P05177 1/20 0.33
CYP3A4 P08684 1/20 0.33
CYP2D6 P10635 1/20 0.33
MAPK1 P28482 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33
AKR1B1 P15121 1/20 0.32
TRPV1 Q8NER1 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15740469 0.88 CYP2C19 (0.34) TMEM97CYP2C19MAPK1NPSR1
SCHEMBL15740440 0.87 KCNH2 (0.36) TMEM97MAPK1NPSR1
SCHEMBL15740437 0.83 MAPK1 (0.38) TMEM97CYP2C19CYP1A2CYP3A4MAPK1
SCHEMBL15740442 0.83 MAPK1 (0.39) TMEM97MAPK1NPSR1
SCHEMBL15740443 0.83 TMEM97 (0.37) TMEM97MAPK1NPSR1
SCHEMBL15740372 0.82 MAPK1 (0.33) MAPK1NPSR1AKR1B1
SCHEMBL15740432 0.82 MAPK1 (0.36) TMEM97MAPK1NPSR1AKR1B1
SCHEMBL15740475 0.82 MAPK1 (0.37) TMEM97CYP2C19CYP1A2CYP3A4MAPK1
SCHEMBL15740499 0.80 TMEM97 (0.40) TMEM97
SCHEMBL15740408 0.80 PTGES (0.38) TMEM97CYP2C19CYP1A2CYP3A4CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2922845-A2 ANTHELMINTIC COMPOUNDS AND COMPOSITIONS AND METHOD OF USING THEREOF Merial, Inc. (US) 2015-09-30 EP disclosed
WO-2014081697-A2 ANTHELMINTIC COMPOUNDS AND COMPOSITIONS AND METHOD OF USING THEREOF MERIAL LIMITED (US) 2014-05-30 WO disclosed