SCHEMBL1574443

SCHEMBL1574443

CCCNC(=O)N1CC(N(C(C)C)C(C)C)C1

nearest known ligand 0.44

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
LMNA P02545 1/20 0.44
KMT2A Q03164 6/20 0.41
NPSR1 Q6W5P4 1/20 0.38
TDP1 Q9NUW8 1/20 0.38
CYP2C19 P33261 2/20 0.37
HTT P42858 1/20 0.36
CHRNB2 P17787 1/20 0.36
CHRNB4 P30926 1/20 0.36
CHRNA3 P32297 1/20 0.36
CHRNA4 P43681 1/20 0.36
MEN1 O00255 4/20 0.35
CYP2C9 P11712 1/20 0.34
NAMPT P43490 3/20 0.33
CNR1 P21554 1/20 0.33
CNR2 P34972 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1574642 0.88 NAMPT (0.48) TDP1HTTNAMPT
SCHEMBL1574970 0.81 LMNA (0.43) LMNAKMT2ANPSR1TDP1CYP2C19
SCHEMBL1574449 0.80 LMNA (0.47) LMNAKMT2ANPSR1TDP1CYP2C19
SCHEMBL1574649 0.79 LMNA (0.46) LMNAKMT2ANPSR1TDP1CYP2C19
SCHEMBL1574751 0.78 ALDH1A1 (0.48) KMT2ANPSR1CYP2C19MEN1CYP2C9
SCHEMBL1574915 0.74 ADAM17 (0.50) HTTNAMPT
SCHEMBL1575097 0.74 KDM4E (0.52) KMT2ANPSR1MEN1
SCHEMBL25853767 0.71 LMNA (0.48) LMNAKMT2ANPSR1CYP2C19HTT
SCHEMBL25849283 0.71 LMNA (0.48) LMNAKMT2ANPSR1CYP2C19HTT
SCHEMBL4089086 0.71 LMNA (0.51) LMNAKMT2ANPSR1TDP1CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2308562-A2 Azetidine ring compounds and drugs comprising the same Ono Pharmaceutical Co., Ltd. (JP) 2011-04-13 EP disclosed
US-7511159-B2 Azetidine ring compounds and drugs comprising the same ONO PHARMACEUTICAL CO., LTD. (JP) 2009-03-31 US disclosed
US-20070135402-A1 Azetidine ring compounds and drugs comprising the same ONO PHARMACEUTICAL CO., LTD. (JP) 2007-06-14 US disclosed
EP-1698375-A1 AZETIDINE RING COMPOUNDS AND DRUGS COMPRISING THE SAME ONO PHARMACEUTICAL CO., LTD. (JP) 2006-09-06 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070135402-A1 Azetidine ring compounds and drugs comprising the same EDNRA, LIPG, EDNRB LMNA 1076/4885KMT2A 2539/4885NPSR1 1387/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.