SCHEMBL15775238

SCHEMBL15775238

Cc1cccc2c1CC(c1ccncc1)=NC2=O

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP10 Q53GL7 2/20 0.39
PARP11 Q9NR21 2/20 0.39
PARP1 P09874 1/20 0.39
MAPK14 Q16539 1/20 0.36
ACHE P22303 1/20 0.36
CDK5 Q00535 1/20 0.36
CDK5R1 Q15078 1/20 0.36
CYP3A4 P08684 1/20 0.36
GRM2 Q14416 1/20 0.35
CYP46A1 Q9Y6A2 1/20 0.34
MAOA P21397 1/20 0.34
CYP19A1 P11511 6/20 0.33
GCGR P47871 1/20 0.33
MGAM O43451 1/20 0.33
GAA P10253 1/20 0.33
SI P14410 1/20 0.33
MGAM2 Q2M2H8 1/20 0.33
IDO1 P14902 1/20 0.33
TYR P14679 1/20 0.33
CYP11B1 P15538 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15775397 0.88 ACHE (0.40) PARP10PARP11PARP1ACHEMAOA
SCHEMBL15775398 0.87 RAB9A (0.40) PARP10PARP11PARP1ACHETYR
SCHEMBL15775414 0.84 SMN1; SMN2 (0.38) PARP10PARP11PARP1ACHEMAOA
SCHEMBL15776267 0.84 NOTUM (0.39) PARP10PARP11PARP1ACHEMGAM
SCHEMBL15775785 0.83 TNKS (0.41) PARP1CYP3A4GRM2MAOA
SCHEMBL15775739 0.82 TNKS (0.40) PARP1GAA
SCHEMBL15775471 0.82 PDCD1 (0.35) PARP10PARP11PARP1ACHEGAA
SCHEMBL15775159 0.82 PARP1 (0.36) PARP10PARP11PARP1ACHE
SCHEMBL15775566 0.80 KCNH2 (0.35) ACHECYP3A4
SCHEMBL15775815 0.79 GRM2 (0.40) GRM2MGAMGAASIMGAM2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2014087165-A1 TANKYRASE INHIBITORS UNIVERSITY OF BATH (GB) 2014-06-12 WO claimed
WO-2014087165-A1 TANKYRASE INHIBITORS UNIVERSITY OF BATH (GB) 2014-06-12 WO disclosed