SCHEMBL15775397

SCHEMBL15775397

Cc1cccc2c1CC(c1ccccc1)=NC2=O

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ACHE P22303 2/20 0.40
RAB9A P51151 4/20 0.39
SMN1; SMN2 Q16637 3/20 0.39
ALDH1A1 P00352 4/20 0.38
PARP1 P09874 1/20 0.37
PARP10 Q53GL7 1/20 0.37
PARP11 Q9NR21 1/20 0.37
ADORA3 P0DMS8 1/20 0.37
ADORA2A P29274 1/20 0.37
ADORA1 P30542 1/20 0.37
AXL P30530 1/20 0.37
NPC1 O15118 5/20 0.35
TSHR P16473 2/20 0.35
HPGD P15428 1/20 0.35
KDM4E B2RXH2 2/20 0.35
MAPT P10636 5/20 0.35
TDP1 Q9NUW8 2/20 0.35
KMT2A Q03164 2/20 0.35
GAA P10253 1/20 0.35
PKM P14618 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15775398 0.89 RAB9A (0.40) ACHERAB9ASMN1; SMN2ALDH1A1PARP1
SCHEMBL15775238 0.88 PARP10 (0.39) ACHEPARP1PARP10PARP11GAA
SCHEMBL15775566 0.88 KCNH2 (0.35) ACHERAB9ASMN1; SMN2ALDH1A1NPC1
SCHEMBL15775414 0.87 SMN1; SMN2 (0.38) ACHERAB9ASMN1; SMN2ALDH1A1PARP1
SCHEMBL15776267 0.87 NOTUM (0.39) ACHERAB9ASMN1; SMN2ALDH1A1PARP1
SCHEMBL15775815 0.84 GRM2 (0.40) KDM4EMAPTKMT2AGAAMAOB
SCHEMBL15775159 0.84 PARP1 (0.36) ACHERAB9ASMN1; SMN2ALDH1A1PARP1
SCHEMBL15775739 0.84 TNKS (0.40) RAB9ASMN1; SMN2ALDH1A1PARP1NPC1
SCHEMBL15775785 0.83 TNKS (0.41) PARP1MAPTMAOAMAOB
SCHEMBL15775467 0.82 ALDH1A1 (0.36) RAB9ASMN1; SMN2ALDH1A1ADORA2AADORA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2014087165-A1 TANKYRASE INHIBITORS UNIVERSITY OF BATH (GB) 2014-06-12 WO claimed
WO-2014087165-A1 TANKYRASE INHIBITORS UNIVERSITY OF BATH (GB) 2014-06-12 WO disclosed