SCHEMBL15775400

SCHEMBL15775400

CCc1cccc2c1CC(c1ccc(CN3CCCCC3)cc1)=NC2=O

nearest known ligand 0.47

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 1/20 0.47
CYP2C19 P33261 1/20 0.47
HRH3 Q9Y5N1 13/20 0.43
HRH4 Q9H3N8 1/20 0.43
OPRM1 P35372 1/20 0.41
OPRK1 P41145 1/20 0.41
DCTPP1 Q9H773 2/20 0.41
PARP1 P09874 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15775445 0.88 CYP2D6 (0.48) CYP2D6CYP2C19HRH3HRH4OPRM1
SCHEMBL15775245 0.86 CYP2D6 (0.46) CYP2D6CYP2C19HRH3HRH4OPRM1
Hydrochloric Acid SCHEMBL15775376 0.85 CYP2D6 (0.45) CYP2D6CYP2C19HRH3HRH4OPRM1
SCHEMBL15775467 0.79 ALDH1A1 (0.36) CYP2D6CYP2C19
SCHEMBL155167 0.65 HRH3 (0.78) CYP2D6CYP2C19HRH3HRH4
SCHEMBL15775399 0.65 TNKS (0.63) CYP2D6CYP2C19HRH3HRH4PARP1
SCHEMBL15775398 0.65 RAB9A (0.40) PARP1
Hydrochloric Acid SCHEMBL7406183 0.64 HRH3 (0.75) CYP2D6CYP2C19HRH3HRH4
Bromide SCHEMBL15775273 0.64 MAOA (0.35) PARP1
SCHEMBL8244456 0.64 HRH3 (0.74) CYP2D6CYP2C19HRH3HRH4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2014087165-A1 TANKYRASE INHIBITORS UNIVERSITY OF BATH (GB) 2014-06-12 WO disclosed