SCHEMBL15775445

SCHEMBL15775445

Cc1cccc2c1CC(c1ccc(CN3CCCCC3)cc1)=NC2=O

nearest known ligand 0.48

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 1/20 0.48
CYP2C19 P33261 1/20 0.48
HRH3 Q9Y5N1 9/20 0.44
HRH4 Q9H3N8 1/20 0.44
DCTPP1 Q9H773 2/20 0.43
OPRM1 P35372 1/20 0.42
OPRK1 P41145 1/20 0.42
PARP1 P09874 2/20 0.41
PTAFR P25105 1/20 0.40
MAPT P10636 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15775245 0.99 CYP2D6 (0.46) CYP2D6CYP2C19HRH3HRH4DCTPP1
Hydrochloric Acid SCHEMBL15775376 0.98 CYP2D6 (0.45) CYP2D6CYP2C19HRH3HRH4DCTPP1
SCHEMBL15775400 0.88 CYP2D6 (0.47) CYP2D6CYP2C19HRH3HRH4DCTPP1
SCHEMBL15776267 0.79 NOTUM (0.39) CYP2C19PARP1MAPT
SCHEMBL15775398 0.79 RAB9A (0.40) PARP1MAPT
SCHEMBL15775397 0.77 ACHE (0.40) PARP1MAPT
SCHEMBL15775414 0.76 SMN1; SMN2 (0.38) PARP1MAPT
SCHEMBL15775238 0.75 PARP10 (0.39) PARP1
SCHEMBL15775739 0.74 TNKS (0.40) PARP1MAPT
SCHEMBL15775159 0.74 PARP1 (0.36) PARP1PTAFRMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2014087165-A1 TANKYRASE INHIBITORS UNIVERSITY OF BATH (GB) 2014-06-12 WO claimed
WO-2014087165-A1 TANKYRASE INHIBITORS UNIVERSITY OF BATH (GB) 2014-06-12 WO disclosed