SCHEMBL15775482

SCHEMBL15775482

Nc1ccc(-c2nc(=O)c3cccc(O)c3[nH]2)cc1

nearest known ligand 0.63

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 15/20 0.63
TNKS O95271 14/20 0.63
TNKS2 Q9H2K2 14/20 0.63
NPC1 O15118 2/20 0.42
POLB P06746 2/20 0.42
RAB9A P51151 2/20 0.42
MEN1 O00255 1/20 0.42
KMT2A Q03164 1/20 0.42
KDM4E B2RXH2 1/20 0.41
ALDH1A1 P00352 1/20 0.41
TP53 P04637 1/20 0.41
MAPT P10636 1/20 0.41
HPGD P15428 1/20 0.41
GFER P55789 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
HSD17B10 Q99714 1/20 0.41
GUSB P08236 1/20 0.40
ADORA2B P29275 1/20 0.40
ADORA1 P30542 1/20 0.40
EGFR P00533 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15775567 0.88 PARP1 (0.61) PARP1TNKSTNKS2KDM4EGUSB
SCHEMBL15775644 0.87 TNKS (0.60) PARP1TNKSTNKS2KDM4EGUSB
SCHEMBL15775241 0.86 TNKS (0.63) PARP1TNKSTNKS2TP53MAPT
SCHEMBL15775381 0.86 TNKS (0.63) PARP1TNKSTNKS2NPC1RAB9A
SCHEMBL15775691 0.86 TNKS (0.63) PARP1TNKSTNKS2KDM4E
SCHEMBL15775320 0.86 TNKS (0.63) PARP1TNKSTNKS2GUSBEGFR
SCHEMBL15775690 0.83 TNKS (0.63) PARP1TNKSTNKS2NPC1POLB
SCHEMBL15775430 0.82 TNKS (0.65) PARP1TNKSTNKS2RAB9A
SCHEMBL1387250 0.81 TNKS (0.66) PARP1TNKSTNKS2NPC1RAB9A
SCHEMBL15775271 0.80 TNKS (0.65) PARP1TNKSTNKS2POLBMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2014087165-A1 TANKYRASE INHIBITORS UNIVERSITY OF BATH (GB) 2014-06-12 WO disclosed