SCHEMBL27639739

SCHEMBL27639739

NC(=O)NSc1ccc(Oc2ccccc2)cc1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP10 Q53GL7 2/20 0.53
SMN1; SMN2 Q16637 3/20 0.44
HPGD P15428 1/20 0.44
PGR P06401 1/20 0.44
ALDH1A1 P00352 2/20 0.43
SRD5A2 P31213 1/20 0.43
SCN4A P35499 1/20 0.43
ERCC5 P28715 1/20 0.42
FEN1 P39748 1/20 0.42
LTA4H P09960 2/20 0.42
NR1H2 P55055 1/20 0.42
BAX Q07812 1/20 0.42
MAOA P21397 1/20 0.42
TGM2 P21980 2/20 0.42
F13A1 P00488 1/20 0.42
CTNNB1 P35222 1/20 0.42
RNF4 P78317 1/20 0.41
TSHR P16473 1/20 0.41
KMT2A Q03164 1/20 0.41
PARP15 Q460N3 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL158241 0.83 SIRT1 (0.42) SMN1; SMN2HPGDALDH1A1TSHRKMT2A
SCHEMBL27946068 0.82 LTA4H (0.47) PARP10SMN1; SMN2HPGDALDH1A1LTA4H
SCHEMBL27798844 0.81 OPRM1 (0.46) LTA4H
SCHEMBL4558245 0.80 NPC1 (0.41) SMN1; SMN2ERCC5FEN1TSHR
SCHEMBL9536223 0.80 PARP10 (0.59) PARP10SMN1; SMN2SRD5A2LTA4HMAOA
SCHEMBL27798703 0.80 KMT2A (0.54) SMN1; SMN2ALDH1A1SRD5A2SCN4AF13A1
SCHEMBL27527894 0.79 CA1 (0.50) PARP10SMN1; SMN2PARP4
Dimethylamine SCHEMBL27576834 0.78 LMNA (0.40) SMN1; SMN2HPGDALDH1A1TSHRKMT2A
SCHEMBL28861802 0.77 CTNNB1 (0.51) PARP10SMN1; SMN2CTNNB1TSHRKMT2A
SCHEMBL5528839 0.76 TRPA1 (0.47) SMN1; SMN2HPGDALDH1A1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101687816-A Triaminopyrimidine derivatives as the CDC25 inhibitors of phosphatases IPSEN PHARMA SAS 2010-03-31 CN claimed
CN-1849301-A Substituted arylthiourea derivatives useful as inhibitors of viral replication ACHILLION PHARMACEUTICALS INC (US) 2006-10-18 CN claimed
CN-107629022-A A kind of Trimethoprim and its preparation method and purposes 上海医药工业研究院 2018-01-26 CN disclosed
CN-107235916-A A kind of licochalcone A deracil analog derivative and its synthetic method for having antitumor activity 陕西科技大学 2017-10-10 CN disclosed
CN-101687816-A Triaminopyrimidine derivatives as the CDC25 inhibitors of phosphatases IPSEN PHARMA SAS 2010-03-31 CN disclosed