SCHEMBL15849166

SCHEMBL15849166

CC(C)[C@@H]1Cc2cc(Br)c(O)cc2CCN1C(=O)C(F)(F)F

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 8/20 0.41
ESR2 Q92731 8/20 0.41
MTNR1B P49286 1/20 0.35
CA12 O43570 1/20 0.33
CA1 P00915 1/20 0.33
CA2 P00918 1/20 0.33
CA7 P43166 1/20 0.33
CA9 Q16790 1/20 0.33
DRD1 P21728 5/20 0.32
DRD5 P21918 2/20 0.32
DRD2 P14416 2/20 0.32
CYP1A2 P05177 1/20 0.32
CYP2D6 P10635 1/20 0.32
TSHR P16473 1/20 0.32
CYP2C19 P33261 1/20 0.32
HSD17B10 Q99714 1/20 0.32
ADCY2 Q08462 1/20 0.32
LMNA P02545 1/20 0.32
ADRA2A P08913 1/20 0.32
ADRA2B P18089 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15849139 0.83 ESR1 (0.37) ESR1ESR2MTNR1BCA12CA1
SCHEMBL15828479 0.76 ESR1 (0.55) ESR1ESR2CA12CA1CA2
SCHEMBL6631121 0.72 ESR1 (0.41) ESR1ESR2MTNR1BCA12CA1
SCHEMBL17890603 0.72 ESR1 (0.62) ESR1ESR2CA12CA1CA2
SCHEMBL1094997 0.72 ESR1 (0.41) ESR1ESR2DRD1DRD5DRD2
SCHEMBL18408135 0.68 HSD11B1 (0.47) ESR1ESR2
SCHEMBL6631355 0.68 MTNR1B (0.46) ESR1ESR2MTNR1BTSHRLMNA
SCHEMBL18407969 0.67 SIGMAR1 (0.57)
SCHEMBL1396472 0.67 SIGMAR1 (0.57)
SCHEMBL1207171 0.67 SIGMAR1 (0.57)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8765780-B2 Alicyclic carboxylic acid derivatives of benzomorphans and related scaffolds, medicaments containing such compounds and their use BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2014-07-01 US disclosed