SCHEMBL15903443

SCHEMBL15903443

Nc1cc(Cl)c(F)c(C(=O)C2CC2)c1

nearest known ligand 0.36

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
TYK2 P29597 1/20 0.36
HSD11B1 P28845 3/20 0.35
THRB P10828 1/20 0.35
HPGD P15428 2/20 0.34
MELK Q14680 4/20 0.33
ALDH1A1 P00352 3/20 0.33
CYP3A4 P08684 1/20 0.33
BACE1 P56817 1/20 0.33
MGLL Q99685 2/20 0.33
KMT2A Q03164 2/20 0.33
MEN1 O00255 1/20 0.32
TSHR P16473 1/20 0.32
NPSR1 Q6W5P4 1/20 0.32
NPC1 O15118 1/20 0.32
RAB9A P51151 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20045609 0.77 TDP1 (0.46) THRBHPGDALDH1A1CYP3A4KMT2A
SCHEMBL15905413 0.74 RORC (0.44) TYK2HPGDALDH1A1KMT2AMEN1
SCHEMBL1029756 0.69 CYP3A4 (0.58) THRBHPGDALDH1A1CYP3A4BACE1
SCHEMBL30606587 0.68 KDM2B (0.46) HSD11B1HPGDMGLLKMT2ATSHR
SCHEMBL26599052 0.68 KDM2B (0.46) HSD11B1HPGDMGLLKMT2ATSHR
SCHEMBL23580096 0.67 TYK2 (0.39) TYK2HSD11B1MELKCYP3A4MGLL
SCHEMBL30461435 0.67 HPGD (0.42) HPGDMELKALDH1A1MGLLKMT2A
SCHEMBL25253119 0.67 HPGD (0.42) HPGDMELKALDH1A1MGLLKMT2A
SCHEMBL12202677 0.66 SMN1; SMN2 (0.44) HSD11B1HPGDALDH1A1MGLLKMT2A
Hydrochloric Acid SCHEMBL30461452 0.66 HPGD (0.41) HPGDMELKALDH1A1MGLLKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 31 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2948149-B1 TOXIC ALDEHYDE RELATED DISEASES AND TREATMENT ALDEYRA THERAPEUTICS INC (US) 2026-03-04 EP disclosed
US-20250127733-A1 TOXIC ALDEHYDE RELATED DISEASES AND TREATMENT ALDEYRA THERAPEUTICS, INC. 2025-04-24 US disclosed
US-20240189260-A1 TOXIC ALDEHYDE RELATED DISEASES AND TREATMENT ALDEYRA THERAPEUTICS, INC. 2024-06-13 US disclosed
CN-117045653-A Diseases and treatments associated with toxic aldehydes 奥尔德拉医疗公司 2023-11-14 CN disclosed
US-11771664-B2 Toxic aldehyde related diseases and treatment ALDEYRA THERAPEUTICS, INC. (US) 2023-10-03 US disclosed
CN-111135171-B Diseases and treatments associated with toxic aldehydes 奥尔德拉医疗公司 2023-09-08 CN disclosed
US-11701331-B2 Toxic aldehyde related diseases and treatment ALDEYRA THERAPEUTICS, INC. (US) 2023-07-18 US disclosed
US-20220354857-A1 ALDEHYDE CONJUGATES AND USES THEREOF ALDEYRA THERAPEUTICS, INC. 2022-11-10 US disclosed
US-20220202745-A1 TOXIC ALDEHYDE RELATED DISEASES AND TREATMENT ALDEYRA THERAPEUTICS, INC. 2022-06-30 US disclosed
CN-114085236-A Aldehyde conjugates and uses thereof 奥尔德拉医疗公司 2022-02-25 CN disclosed
EP-3337470-A1 ALDEHYDE CONJUGATES AND USES THEREOF Aldeyra Therapeutics, Inc. (US) 2018-06-27 EP disclosed
US-20170239196-A1 TOXIC ALDEHYDE RELATED DISEASES AND TREATMENT ALDEYRA THERAPEUTICS, INC. (F/K/A ALDEXA THERAPEUTICS, INC. F/K/A NEURON SYSTEMS, INC.) 2017-08-24 US disclosed
US-9687481-B2 Toxic aldehyde related diseases and treatment ALDEYRA THERAPEUTICS, INC. (US) 2017-06-27 US disclosed
WO-2017035082-A1 ALDEHYDE CONJUGATES AND USES THEREOF ALDEYRA THERAPEUTICS, INC. (US) 2017-03-02 WO disclosed
US-20150344447-A1 NOVEL TRAPS IN THE TREATMENT OF MACULAR DEGENERATION ALDEXA THERAPEUTICS, INC. 2015-12-03 US disclosed
EP-2948436-A1 NOVEL TRAPS IN THE TREATMENT OF MACULAR DEGENERATION Aldeyra Therapeutics, Inc. (US) 2015-12-02 EP disclosed
EP-2948149-A2 TOXIC ALDEHYDE RELATED DISEASES AND TREATMENT Aldeyra Therapeutics, Inc. (US) 2015-12-02 EP disclosed
US-20150335632-A1 TOXIC ALDEHYDE RELATED DISEASES AND TREATMENT ALDEYRA THERAPEUTICS, INC. (F/K/A ALDEXA THERAPEUTICS, INC. F/K/A NEURON SYSTEMS, INC.) 2015-11-26 US disclosed
WO-2014116836-A2 TOXIC ALDEHYDE RELATED DISEASES AND TREATMENT ALDEXA THERAPEUTICS, INC. (US) 2014-07-31 WO disclosed
WO-2014116593-A1 NOVEL TRAPS IN THE TREATMENT OF MACULAR DEGENERATION ALDEXA THERAPEUTICS, INC. (US) 2014-07-31 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (9 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20170239196-A1 TOXIC ALDEHYDE RELATED DISEASES AND TREATMENT ALDH1A2, ALDH2, ALDH1A1 TYK2 3739/4885HSD11B1 846/4885THRB 4466/4885
US-20150344447-A1 NOVEL TRAPS IN THE TREATMENT OF MACULAR DEGENERATION PDE6C, PDE6D, PDE6A TYK2 4567/4885HSD11B1 1313/4885THRB 2028/4885
US-20250127733-A1 TOXIC ALDEHYDE RELATED DISEASES AND TREATMENT ALDH1A2, ALDH2, ALDH1A1 TYK2 3739/4885HSD11B1 846/4885THRB 4466/4885
US-11771664-B2 Toxic aldehyde related diseases and treatment ALDH1A2, ALDH2, ALDH1A1 TYK2 3739/4885HSD11B1 846/4885THRB 4466/4885
US-11701331-B2 Toxic aldehyde related diseases and treatment ALDH1A2, ALDH2, ALDH1A1 TYK2 3739/4885HSD11B1 846/4885THRB 4466/4885
US-20220202745-A1 TOXIC ALDEHYDE RELATED DISEASES AND TREATMENT ALDH1A2, ALDH2, ALDH1A1 TYK2 3739/4885HSD11B1 846/4885THRB 4466/4885
US-20150335632-A1 TOXIC ALDEHYDE RELATED DISEASES AND TREATMENT ALDH1A2, ALDH2, ALDH1A1 TYK2 3739/4885HSD11B1 846/4885THRB 4466/4885
US-20220354857-A1 ALDEHYDE CONJUGATES AND USES THEREOF ALDH1A2, AOX1, ALDH2 TYK2 2800/4885HSD11B1 1223/4885THRB 4627/4885
US-20240189260-A1 TOXIC ALDEHYDE RELATED DISEASES AND TREATMENT ALDH1A2, ALDH2, ALDH1A1 TYK2 3739/4885HSD11B1 846/4885THRB 4466/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.