SCHEMBL1865507

SCHEMBL1865507

c1ccc(C2(c3cccnc3)CC[N]2)cc1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.42
LMNA P02545 1/20 0.42
OPRM1 P35372 2/20 0.40
OPRL1 P41146 2/20 0.40
MEN1 O00255 2/20 0.40
KMT2A Q03164 2/20 0.40
VNN1 O95497 1/20 0.40
OPRD1 P41143 1/20 0.39
OPRK1 P41145 1/20 0.39
CFTR P13569 1/20 0.37
SLC6A2 P23975 1/20 0.37
SLC6A4 P31645 1/20 0.37
SLC6A3 Q01959 1/20 0.37
GOPC Q9HD26 1/20 0.37
CYP11B1 P15538 1/20 0.37
CYP11B2 P19099 1/20 0.37
HCAR2 Q8TDS4 1/20 0.37
CYP3A4 P08684 1/20 0.37
CHRM2 P08172 1/20 0.36
CHRM4 P08173 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1866642 0.91 ALDH1A1 (0.40) ALDH1A1LMNAOPRM1OPRL1MEN1
SCHEMBL1862411 0.91 ALDH1A1 (0.40) ALDH1A1LMNAOPRM1OPRL1MEN1
SCHEMBL1862897 0.90 LMNA (0.39) ALDH1A1LMNAOPRM1OPRL1MEN1
SCHEMBL1860147 0.80 HTR2A (0.38) ALDH1A1LMNAOPRM1OPRL1MEN1
SCHEMBL1866073 0.80 HTR2A (0.38) ALDH1A1LMNAOPRM1OPRL1MEN1
SCHEMBL1865938 0.80 HTR2A (0.38) ALDH1A1LMNAOPRM1OPRL1MEN1
SCHEMBL1863575 0.78 CHRNB2 (0.37) ALDH1A1LMNAMEN1KMT2ACYP3A4
SCHEMBL159063 0.76 HCAR2 (0.38) ALDH1A1LMNAOPRM1OPRL1MEN1
SCHEMBL9639574 0.72 DPP4 (0.41) LMNAOPRM1OPRD1SLC6A2SLC6A4
SCHEMBL27426615 0.70 ALDH1A1 (0.40) ALDH1A1LMNAOPRM1OPRL1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2493877-A1 PYRIMIDINE COMPOUNDS AS DELTA OPIOID RECEPTOR MODULATORS Janssen Pharmaceutica NV (BE) 2012-09-05 EP disclosed
WO-2011053705-A1 PYRIMIDINE COMPOUNDS AS DELTA OPIOID RECEPTOR MODULATORS JANSSEN PHARMACEUTICA NV (BE) 2011-05-05 WO disclosed