SCHEMBL15933477

SCHEMBL15933477

CC(C)(C)OC(=O)N1CCn2nc(-c3ccc(F)nc3)nc2C1

nearest known ligand 0.40

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
HDAC4 P56524 1/20 0.40
CKS1B P61024 2/20 0.40
SKP1 P63208 2/20 0.40
SKP2 Q13309 2/20 0.40
HDAC8 Q9BY41 1/20 0.39
HDAC6 Q9UBN7 1/20 0.39
GPR119 Q8TDV5 7/20 0.39
GRIA1 P42261 1/20 0.38
DPP4 P27487 1/20 0.38
DPP8 Q6V1X1 1/20 0.38
DPP7 Q9UHL4 1/20 0.38
ESR2 Q92731 1/20 0.38
GBA1 P04062 1/20 0.38
LIPG Q9Y5X9 1/20 0.37
DYRK2 Q92630 1/20 0.37
JAK2 O60674 1/20 0.37
JAK1 P23458 1/20 0.37
NR1H2 P55055 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15933677 0.85 GPR119 (0.53) CKS1BSKP1SKP2GPR119JAK2
SCHEMBL31612680 0.83 HDAC4 (0.48) HDAC4HDAC6GPR119DPP4DPP8
SCHEMBL17984905 0.83 ESR2 (0.40) HDAC4CKS1BSKP1SKP2HDAC6
SCHEMBL20140942 0.82 CKS1B (0.49) HDAC4CKS1BSKP1SKP2GPR119
SCHEMBL15933643 0.81 GPR119 (0.45) HDAC4CKS1BSKP1SKP2GPR119
SCHEMBL15933697 0.81 GPR119 (0.47) HDAC4CKS1BSKP1SKP2GPR119
SCHEMBL15933678 0.81 CSNK1D (0.43) HDAC4CKS1BSKP1SKP2GPR119
SCHEMBL24689567 0.80 NR1H2 (0.43) HDAC4GPR119DPP4DPP8DPP7
SCHEMBL15933535 0.80 GPR119 (0.49) HDAC4GPR119ESR2JAK2JAK1
SCHEMBL31612664 0.79 MAPT (0.40) HDAC4CKS1BSKP1SKP2HDAC8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2014117318-A1 NOVEL TRIAZOLE ANTIFUNGAL COMPOUNDS, AND PHARMACEUTICAL COMPOSITION, PREPARATION METHOD, AND APPLICATION THEREOF 中国科学院上海药物研究所 (CN) 2014-08-07 WO disclosed