SCHEMBL15933535

SCHEMBL15933535

CC(C)(C)OC(=O)N1CCn2nc(-c3ccc(C#N)cc3)nc2C1

nearest known ligand 0.49

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
GPR119 Q8TDV5 8/20 0.49
EGLN2 Q96KS0 3/20 0.46
CSNK1D P48730 1/20 0.42
CSNK1E P49674 1/20 0.42
JAK2 O60674 2/20 0.42
JAK3 P52333 1/20 0.42
PTK2 Q05397 1/20 0.42
HDAC4 P56524 1/20 0.41
PGGT1B P53609 1/20 0.39
JAK1 P23458 1/20 0.39
CETP P11597 1/20 0.39
ESR2 Q92731 1/20 0.38
IRAK4 Q9NWZ3 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15933683 0.87 GPR119 (0.52) GPR119EGLN2PGGT1BCETPESR2
SCHEMBL15933677 0.86 GPR119 (0.53) GPR119EGLN2JAK2JAK1
SCHEMBL20140942 0.85 CKS1B (0.49) GPR119JAK2JAK3HDAC4ESR2
SCHEMBL15933697 0.84 GPR119 (0.47) GPR119HDAC4ESR2
SCHEMBL31612680 0.84 HDAC4 (0.48) GPR119HDAC4ESR2
SCHEMBL24689567 0.83 NR1H2 (0.43) GPR119HDAC4ESR2
SCHEMBL15933643 0.80 GPR119 (0.45) GPR119CSNK1DCSNK1EHDAC4ESR2
SCHEMBL15933477 0.80 HDAC4 (0.40) GPR119JAK2HDAC4JAK1ESR2
SCHEMBL25431827 0.79 GPR119 (0.43) GPR119ESR2
SCHEMBL17984905 0.79 ESR2 (0.40) CSNK1EJAK2HDAC4JAK1ESR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2014117318-A1 NOVEL TRIAZOLE ANTIFUNGAL COMPOUNDS, AND PHARMACEUTICAL COMPOSITION, PREPARATION METHOD, AND APPLICATION THEREOF 中国科学院上海药物研究所 (CN) 2014-08-07 WO disclosed