SCHEMBL15933643

SCHEMBL15933643

CC(C)(C)OC(=O)N1CCn2nc(-c3cncnc3)nc2C1

nearest known ligand 0.45

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
GPR119 Q8TDV5 4/20 0.45
CYP3A4 P08684 1/20 0.40
CYP3A5 P20815 1/20 0.40
GBA1 P04062 1/20 0.40
CKS1B P61024 2/20 0.39
SKP1 P63208 2/20 0.39
SKP2 Q13309 2/20 0.39
ESR2 Q92731 1/20 0.39
CSNK1D P48730 1/20 0.39
CSNK1E P49674 1/20 0.39
NR1H2 P55055 1/20 0.37
MAPT P10636 2/20 0.37
HDAC4 P56524 1/20 0.37
KIT P10721 1/20 0.37
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36
ALDH1A1 P00352 1/20 0.36
LMNA P02545 1/20 0.36
MAPK1 P28482 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15933697 0.86 GPR119 (0.47) GPR119GBA1CKS1BSKP1SKP2
SCHEMBL15933678 0.86 CSNK1D (0.43) GPR119CYP3A4CYP3A5GBA1CKS1B
SCHEMBL20140942 0.85 CKS1B (0.49) GPR119GBA1CKS1BSKP1SKP2
SCHEMBL15933683 0.84 GPR119 (0.52) GPR119GBA1ESR2
SCHEMBL17984905 0.83 ESR2 (0.40) CYP3A4CYP3A5CKS1BSKP1SKP2
SCHEMBL15933477 0.81 HDAC4 (0.40) GPR119GBA1CKS1BSKP1SKP2
SCHEMBL31612680 0.81 HDAC4 (0.48) GPR119ESR2MAPTHDAC4ALDH1A1
SCHEMBL24689567 0.80 NR1H2 (0.43) GPR119ESR2NR1H2HDAC4MEN1
SCHEMBL15933535 0.80 GPR119 (0.49) GPR119ESR2CSNK1DCSNK1EHDAC4
SCHEMBL15933677 0.79 GPR119 (0.53) GPR119CKS1BSKP1SKP2NR1H2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2014117318-A1 NOVEL TRIAZOLE ANTIFUNGAL COMPOUNDS, AND PHARMACEUTICAL COMPOSITION, PREPARATION METHOD, AND APPLICATION THEREOF 中国科学院上海药物研究所 (CN) 2014-08-07 WO disclosed