SCHEMBL15958645

SCHEMBL15958645

COc1nc2ccccc2nc1/C=C/c1ccc(N(C)C)cc1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 7/20 0.52
MEN1 O00255 5/20 0.52
KMT2A Q03164 5/20 0.52
RAB9A P51151 4/20 0.52
KDM4E B2RXH2 1/20 0.52
MAPK1 P28482 1/20 0.52
RXFP1 Q9HBX9 1/20 0.52
L3MBTL1 Q9Y468 1/20 0.52
RELA Q04206 1/20 0.51
APP P05067 8/20 0.50
SMN1; SMN2 Q16637 3/20 0.50
S100A4 P26447 1/20 0.50
INSR P06213 1/20 0.50
NCOA1 Q15788 1/20 0.50
NPC1 O15118 2/20 0.49
ALOX15 P16050 1/20 0.49
CASP1 P29466 1/20 0.49
HBB P68871 1/20 0.49
NQO2 P16083 1/20 0.47
KLF5 Q13887 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10435447 0.86 RELA (0.63) MAPTMEN1KMT2ARAB9AKDM4E
SCHEMBL10371974 0.86 RELA (0.63) MAPTMEN1KMT2ARAB9AKDM4E
SCHEMBL12676802 0.85 S100A4 (0.50) MAPTMEN1KMT2ARAB9AKDM4E
SCHEMBL12669913 0.85 MAPT (0.49) MAPTMEN1KMT2ARAB9AKDM4E
SCHEMBL8219137 0.85 KDM4E (0.48) MAPTMEN1KMT2ARAB9AKDM4E
SCHEMBL8226827 0.84 TRPA1 (0.56) MAPTRAB9AKDM4EL3MBTL1RELA
SCHEMBL14619409 0.79 MAPT (0.55) MAPTMEN1KMT2ARAB9AKDM4E
SCHEMBL10435351 0.77 APP (0.61) MAPTMEN1KMT2ARAB9AKDM4E
SCHEMBL8224935 0.75 CYP11B1 (0.53) MEN1KMT2ARAB9AKDM4ESMN1; SMN2
SCHEMBL30464972 0.75 MAPT (0.61) MAPTMEN1KMT2ARAB9AKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8809264-B2 Quinoxalinyl macrocyclic hepatitis C virus serine protease inhibitors ENANTA PHARMACEUTICALS, INC. (US) 2014-08-19 US disclosed