SCHEMBL15958950

SCHEMBL15958950

CCC(=O)c1cccc(O)c1N

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
G6PD P11413 1/20 0.60
CASP7 P55210 1/20 0.60
CASP6 P55212 1/20 0.60
KDM4E B2RXH2 4/20 0.58
HIF1A Q16665 1/20 0.58
TDP1 Q9NUW8 1/20 0.58
HSP90AB1 P08238 1/20 0.47
MAPT P10636 3/20 0.41
ALDH1A1 P00352 3/20 0.41
HPGD P15428 2/20 0.41
TSHR P16473 1/20 0.41
HSD17B10 Q99714 1/20 0.41
HTT P42858 2/20 0.41
HMGCR P04035 1/20 0.41
CA12 O43570 2/20 0.40
CA1 P00915 2/20 0.40
CA2 P00918 2/20 0.40
CA7 P43166 2/20 0.40
CA9 Q16790 2/20 0.40
CA14 Q9ULX7 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10970621 0.88 HSP90AB1 (0.44) G6PDCASP7CASP6KDM4EHIF1A
SCHEMBL9632452 0.82 ALDH1A1 (0.46) G6PDCASP7CASP6KDM4EHIF1A
SCHEMBL9058909 0.81 GABRA1 (0.43) KDM4EHIF1ATDP1HSP90AB1ALDH1A1
SCHEMBL7547028 0.81 CD44 (0.43) G6PDCASP7CASP6KDM4EHIF1A
SCHEMBL8691817 0.81 PARP1 (0.42) G6PDCASP7CASP6KDM4EHIF1A
SCHEMBL27355845 0.81 G6PD (0.60) G6PDCASP7CASP6KDM4EHIF1A
SCHEMBL14255774 0.80 KDM4E (0.67) G6PDCASP7CASP6KDM4EHIF1A
SCHEMBL17653405 0.80 CTSD (0.49) KDM4EMAPTALDH1A1HPGDHSD17B10
SCHEMBL1606580 0.80 HSP90AB1 (0.55) TDP1HSP90AB1MAPTALDH1A1HPGD
SCHEMBL15153940 0.80 HTT (0.64) G6PDCASP7CASP6KDM4EHIF1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102838505-B Amides, its preparation method and application SHANGHAI INSTITUTE OF PHARMACEUTICAL INDUSTRY (CN) 2016-02-17 CN disclosed
EP-2421825-B9 AZETIDINYL DIAMIDES AS MONOACYLGLYCEROL LIPASE INHIBITORS JANSSEN PHARMACEUTICA NV (BE) 2014-08-20 EP disclosed
EP-2421825-B1 AZETIDINYL DIAMIDES AS MONOACYLGLYCEROL LIPASE INHIBITORS JANSSEN PHARMACEUTICA NV (BE) 2014-01-01 EP disclosed
CN-102838505-A Amide compound and preparation method as well as application thereof SHANGHAI INST PHARM INDUSTRY 2012-12-26 CN disclosed