SCHEMBL15973191

SCHEMBL15973191

Cc1ccccc1CN1CC(=O)NC1=O

nearest known ligand 0.58

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 2/20 0.58
MEN1 O00255 1/20 0.58
SMN1; SMN2 Q16637 1/20 0.58
MAPT P10636 1/20 0.55
P2RX7 Q99572 2/20 0.49
PTGS1 P23219 1/20 0.49
PTGS2 P35354 1/20 0.49
TRPC5 Q9UL62 5/20 0.45
LMNA P02545 1/20 0.45
CYP2A13 Q16696 1/20 0.42
EPHX2 P34913 1/20 0.42
DDB1 Q16531 1/20 0.41
CRBN Q96SW2 1/20 0.41
ACHE P22303 1/20 0.41
KDM4E B2RXH2 1/20 0.41
POLB P06746 1/20 0.41
SIRT2 Q8IXJ6 1/20 0.41
SIRT1 Q96EB6 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9871553 0.81 LMNA (0.58) KMT2AMEN1SMN1; SMN2MAPTP2RX7
SCHEMBL8633466 0.80 CYP1A2 (0.50) KMT2AMEN1SMN1; SMN2MAPTP2RX7
SCHEMBL6938726 0.80 EPHX2 (0.42) KMT2AMEN1SMN1; SMN2MAPTP2RX7
SCHEMBL11570834 0.80 MPO (0.49) EPHX2DDB1CRBNKDM4EPOLB
SCHEMBL7696982 0.80 EPHX2 (0.39) KMT2AMEN1SMN1; SMN2MAPTTRPC5
SCHEMBL877544 0.80 KMT2A (0.57) KMT2AMEN1SMN1; SMN2MAPTP2RX7
SCHEMBL8128225 0.78 DAO (0.48) MAPTACHEPOLB
SCHEMBL4512688 0.75 KMT2A (0.65) KMT2AMEN1SMN1; SMN2MAPTP2RX7
SCHEMBL9850086 0.75 DDB1 (0.69) KMT2AMEN1EPHX2DDB1CRBN
SCHEMBL1011633 0.75 DDB1 (0.69) KMT2AMEN1EPHX2DDB1CRBN

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2958897-A2 COMPOUNDS USEFUL AS MODULATORS OF TRPM8 Senomyx, Inc. (US) 2015-12-30 EP disclosed
WO-2014130582-A2 COMPOUNDS USEFUL AS MODULATORS OF TRPM8 SENOMYX, INC. (US) 2014-08-28 WO disclosed