SCHEMBL1600115

SCHEMBL1600115

COc1cc(-n2nc(C(=O)O)c3ccccc32)c(C(C)(C)C)cc1C(N)=O

nearest known ligand 0.48

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 3/20 0.47
ALDH1A1 P00352 1/20 0.47
SCN9A Q15858 1/20 0.41
MAP3K14 Q99558 9/20 0.41
RORC P51449 1/20 0.40
BCL2 P10415 3/20 0.39
STAT1 P42224 2/20 0.39
MEN1 O00255 2/20 0.37
PKM P14618 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1600053 0.75 SCN9A (0.36) KMT2AALDH1A1SCN9AMAP3K14RORC
SCHEMBL9025523 0.72 RORC (0.56) KMT2AALDH1A1SCN9ARORCSTAT1
SCHEMBL5652361 0.69 PDE10A (0.48) KMT2AALDH1A1RORCSTAT1MEN1
SCHEMBL22949523 0.69 HPGD (0.47) ALDH1A1
SCHEMBL9024249 0.68 ALDH1A1 (0.57) ALDH1A1SCN9ARORCBCL2STAT1
SCHEMBL1600387 0.67 CHRM5 (0.41) KMT2A
SCHEMBL27712242 0.66 F12 (0.59) KMT2A
SCHEMBL27732440 0.65 ELANE (0.56) KMT2AALDH1A1MEN1
SCHEMBL28774901 0.65 ELANE (0.56) KMT2AMEN1PKM
SCHEMBL7421574 0.65 SCN9A (0.58) ALDH1A1SCN9ARORCSTAT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7919617-B2 Cytokine inhibitors iTherX Pharmaceuticals Inc. (US) 2011-04-05 US disclosed
US-7897599-B2 Cytokine inhibitors iTherX Pharmaceuticals Inc. (US) 2011-03-01 US disclosed