SCHEMBL16003992

SCHEMBL16003992

COc1ccc(CCOCc2ccc3c(c2)CN(C(C)=O)CCO3)cc1OC

nearest known ligand 0.45

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 3/20 0.45
MEN1 O00255 2/20 0.45
HTT P42858 2/20 0.44
CHRM5 P08912 5/20 0.44
CHRM1 P11229 5/20 0.44
LMNA P02545 1/20 0.41
CXCR3 P49682 1/20 0.41
ALDH1A1 P00352 2/20 0.41
TSHR P16473 1/20 0.40
CYP2C19 P33261 1/20 0.40
CHRM3 P20309 2/20 0.40
GPR142 Q7Z601 1/20 0.40
CHRM2 P08172 1/20 0.40
CHRM4 P08173 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.39
NTRK1 P04629 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16003986 0.87 ALDH1A1 (0.42) KMT2AMEN1HTTCHRM5CHRM1
SCHEMBL16003985 0.87 ATM (0.43) KMT2AMEN1HTTCHRM5CHRM1
SCHEMBL16003990 0.86 CHRM5 (0.43) KMT2AMEN1HTTCHRM5CHRM1
SCHEMBL16003993 0.85 GAA (0.51) KMT2AMEN1HTTCHRM5CHRM1
SCHEMBL16003994 0.85 GPR142 (0.60) CHRM5CHRM1ALDH1A1GPR142
SCHEMBL16004317 0.78 GPR142 (0.61) KMT2AMEN1CHRM5CHRM1ALDH1A1
SCHEMBL16004254 0.76 PIK3CA (0.47) KMT2AMEN1HTTLMNAALDH1A1
SCHEMBL16004091 0.76 ALDH1A1 (0.48) KMT2AMEN1LMNAALDH1A1GPR142
SCHEMBL16004308 0.73 ABCB1 (0.48) KMT2AMEN1HTTALDH1A1GPR142
SCHEMBL16004303 0.73 HPGD (0.49) KMT2ALMNASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2014133414-A2 HETEROCYCLIC TGR5 BILE ACID RECEPTOR AGONISTS, PHARMACEUTICAL COMPOSITION, METHODS FOR THE PRODUCTION AND USE THEREOF АЛЛА ХЕМ ЛЛС (US) 2014-09-04 WO disclosed