SCHEMBL16003993

SCHEMBL16003993

COc1ccc(CCOCc2ccc3c(c2)CN(C(=O)c2cccs2)CCO3)cc1OC

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 1/20 0.51
ALDH1A1 P00352 4/20 0.44
CYP1A2 P05177 1/20 0.44
CYP2D6 P10635 1/20 0.44
CYP2C9 P11712 1/20 0.44
CYP2C19 P33261 1/20 0.44
LMNA P02545 3/20 0.43
CASP1 P29466 1/20 0.43
CASP7 P55210 1/20 0.43
HSD17B10 Q99714 1/20 0.43
NPSR1 Q6W5P4 1/20 0.42
CHRM5 P08912 2/20 0.41
CHRM1 P11229 2/20 0.41
KDM4E B2RXH2 2/20 0.40
PKM P14618 1/20 0.40
KMT2A Q03164 3/20 0.39
MEN1 O00255 2/20 0.39
RECQL P46063 1/20 0.39
SIRT5 Q9NXA8 1/20 0.39
HTT P42858 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16004095 0.88 LMNA (0.43) GAAALDH1A1LMNACHRM5CHRM1
SCHEMBL16003992 0.85 KMT2A (0.45) ALDH1A1CYP2C19LMNACHRM5CHRM1
SCHEMBL16003990 0.84 CHRM5 (0.43) LMNAHSD17B10CHRM5CHRM1KDM4E
SCHEMBL16003983 0.84 GAA (0.43) GAAALDH1A1CYP1A2CYP2D6CYP2C9
SCHEMBL16003985 0.83 ATM (0.43) GAAALDH1A1CHRM5CHRM1KDM4E
SCHEMBL16003974 0.82 HRH3 (0.52) GAALMNAKMT2A
SCHEMBL16003994 0.80 GPR142 (0.60) ALDH1A1CHRM5CHRM1KDM4EPKM
SCHEMBL16004103 0.80 LMNA (0.44) GAAALDH1A1CYP1A2CYP2D6CYP2C9
SCHEMBL16003986 0.80 ALDH1A1 (0.42) ALDH1A1LMNACHRM5CHRM1KDM4E
SCHEMBL16004143 0.79 LMNA (0.43) GAAALDH1A1CYP2C9LMNAKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2014133414-A2 HETEROCYCLIC TGR5 BILE ACID RECEPTOR AGONISTS, PHARMACEUTICAL COMPOSITION, METHODS FOR THE PRODUCTION AND USE THEREOF АЛЛА ХЕМ ЛЛС (US) 2014-09-04 WO disclosed