SCHEMBL16004232

SCHEMBL16004232

CCC(=O)N(C)Cc1ccc2c(c1)CN(C(=O)c1cccnc1)CCO2

nearest known ligand 0.49

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
PIK3CA P42336 7/20 0.49
KDM4E B2RXH2 2/20 0.46
TDP1 Q9NUW8 2/20 0.46
HPGD P15428 1/20 0.44
RIPK1 Q13546 1/20 0.41
GAA P10253 1/20 0.41
PDGFRB P09619 1/20 0.39
KDR P35968 1/20 0.39
CTNNB1 P35222 1/20 0.39
WNT3A P56704 1/20 0.39
AHR P35869 1/20 0.39
AOC3 Q16853 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16004128 0.86 PIK3CA (0.49) PIK3CAKDM4ETDP1HPGDRIPK1
SCHEMBL16004243 0.83 PIK3CA (0.40) PIK3CAHPGDRIPK1AOC3
SCHEMBL16004271 0.82 RIPK1 (0.45) PIK3CAHPGDRIPK1GAAAOC3
SCHEMBL16004055 0.81 PIK3CA (0.49) PIK3CARIPK1
SCHEMBL16004052 0.80 PIK3CA (0.52) PIK3CAHPGDRIPK1GAAAOC3
SCHEMBL16004283 0.79 CREBBP (0.52)
SCHEMBL16004282 0.77 GPR142 (0.54)
SCHEMBL16004054 0.75 PIK3CA (0.49) PIK3CAHPGDRIPK1AOC3
SCHEMBL16004118 0.75 PIK3CA (0.47) PIK3CARIPK1
SCHEMBL16004274 0.74 RIPK1 (0.46) PIK3CAKDM4EHPGDRIPK1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2014133414-A2 HETEROCYCLIC TGR5 BILE ACID RECEPTOR AGONISTS, PHARMACEUTICAL COMPOSITION, METHODS FOR THE PRODUCTION AND USE THEREOF АЛЛА ХЕМ ЛЛС (US) 2014-09-04 WO disclosed