SCHEMBL16004142

SCHEMBL16004142

COc1cc(C(=O)N2CCOc3ccc(COCc4ccc(C)cc4)cc3C2)cc(OC)c1OC

nearest known ligand 0.47

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
LMNA P02545 1/20 0.44
HTT P42858 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
KDM4E B2RXH2 1/20 0.44
POLB P06746 1/20 0.43
ALDH1A1 P00352 3/20 0.43
CYP1A2 P05177 1/20 0.43
L3MBTL1 Q9Y468 1/20 0.42
ABCB1 P08183 1/20 0.41
RIPK1 Q13546 1/20 0.41
CREBBP Q92793 1/20 0.41
TP53 P04637 1/20 0.40
MAPT P10636 1/20 0.40
NPC1 O15118 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16003982 0.88 ALDH1A1 (0.45) HTTKDM4EPOLBALDH1A1CYP1A2
SCHEMBL16004141 0.79 HTT (0.48) LMNAHTTSMN1; SMN2KDM4EPOLB
SCHEMBL16004247 0.79 HPGD (0.51) LMNASMN1; SMN2POLBALDH1A1RIPK1
SCHEMBL16003980 0.78 FKBP1A (0.53) SMN1; SMN2KDM4EPOLBALDH1A1CYP1A2
SCHEMBL16004106 0.78 GPR142 (0.51) HTTSMN1; SMN2ALDH1A1RIPK1CREBBP
SCHEMBL16004298 0.76 ALDH1A1 (0.49) LMNAHTTSMN1; SMN2KDM4EPOLB
SCHEMBL16004303 0.76 HPGD (0.49) LMNASMN1; SMN2POLBRIPK1MAPT
SCHEMBL16004096 0.75 MAPT (0.55) POLBRIPK1CREBBPTP53MAPT
SCHEMBL16003985 0.74 ATM (0.43) HTTKDM4EALDH1A1RIPK1TP53
SCHEMBL16003988 0.74 PIK3CA (0.46) LMNASMN1; SMN2ALDH1A1RIPK1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2014133414-A2 HETEROCYCLIC TGR5 BILE ACID RECEPTOR AGONISTS, PHARMACEUTICAL COMPOSITION, METHODS FOR THE PRODUCTION AND USE THEREOF АЛЛА ХЕМ ЛЛС (US) 2014-09-04 WO disclosed